SCHEMBL326696

SCHEMBL326696

c1ccc(CN2CCC3(CCc4cccnc43)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.64
TP53 P04637 2/20 0.64
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2D6 P10635 2/20 0.64
TSHR P16473 2/20 0.64
CYP2C19 P33261 2/20 0.64
ALDH1A1 P00352 1/20 0.64
CYP2C9 P11712 1/20 0.64
HTR2A P28223 4/20 0.59
HTR2C P28335 4/20 0.59
HTR2B P41595 4/20 0.59
DRD2 P14416 3/20 0.59
NFKB1 P19838 1/20 0.54
MAPK1 P28482 1/20 0.54
MTOR P42345 1/20 0.54
TMEM97 Q5BJF2 1/20 0.53
MEN1 O00255 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13855275 0.85 SIGMAR1 (0.67) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL8246067 0.85 SIGMAR1 (0.52) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL326697 0.80 SIGMAR1 (0.55) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL466954 0.79 SIGMAR1 (1.00) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL22545216 0.78 SIGMAR1 (0.50) SIGMAR1HTR2AHTR2CHTR2BDRD2
SCHEMBL2517838 0.76 SIGMAR1 (0.54) SIGMAR1HTR2A
SCHEMBL8237648 0.75 SIGMAR1 (0.44) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL6841309 0.74 SIGMAR1 (1.00) SIGMAR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL22520497 0.73 CYP2D6 (0.41) SIGMAR1CYP2D6HTR2AHTR2CHTR2B
SCHEMBL25855001 0.73 CHRM2 (0.41) SIGMAR1TP53CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590955-A1 SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS ABBVIE B.V. (NL) 2013-05-15 EP disclosed
WO-2012004378-A1 SPIRO-CYCLIC AMINE DERIVATIVES AS S1P MODULATORS ABBOTT HEALTHCARE PRODUCTS B.V. (NL) 2012-01-12 WO disclosed