SCHEMBL326856

SCHEMBL326856

CC1(C)c2ccc(O)cc2CCN1C(=O)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.45
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
DRD1 P21728 10/20 0.43
DRD2 P14416 8/20 0.43
DRD5 P21918 7/20 0.43
DRD3 P35462 7/20 0.43
DRD4 P21917 5/20 0.43
ESR2 Q92731 2/20 0.42
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
AKR1C3 P42330 1/20 0.40
HTR2A P28223 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25324704 0.75 DRD2 (0.58) ESR1DRD1DRD2DRD5DRD3
SCHEMBL1189934 0.74 MAPK1 (0.49) MAPK1ALDH1A1HPGD
SCHEMBL16523571 0.72 CA1 (0.61) ESR1GRIN1GRIN2BESR2ALDH1A1
SCHEMBL3056380 0.72 CA1 (0.68) ESR1GRIN1GRIN2BESR2ALDH1A1
SCHEMBL11031260 0.71 HPGD (0.69) ALDH1A1HPGD
SCHEMBL16494462 0.71 HPGD (0.69) ALDH1A1HPGDCA1CA2CA7
SCHEMBL22533944 0.70 NR1H2 (0.42) ESR1DRD1DRD2DRD5MAPK1
SCHEMBL20738485 0.68 NOTUM (0.47) MAPK1ALDH1A1
SCHEMBL20909774 0.68 NOTUM (0.51) ESR1ALDH1A1AKR1C3
SCHEMBL1189233 0.68 MAPK1 (0.43) MAPK1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130190529-A1 Fluorine Radiolabelling Process ISIS INNOVATION LIMITED (GB) 2013-07-25 US disclosed
US-20130190529-A1 Fluorine Radiolabelling Process ISIS INNOVATION LIMITED (GB) 2013-07-25 US disclosed
US-20130190529-A1 Fluorine Radiolabelling Process ISIS INNOVATION LIMITED (GB) 2013-07-25 US disclosed
EP-2590910-A2 FLUORINE RADIOLABELLING PROCESS Isis Innovation Limited (GB) 2013-05-15 EP disclosed
WO-2012004567-A2 FLUORINE RADIOLABELLING PROCESS ISIS INNOVATION LIMITED (GB) 2012-01-12 WO disclosed
WO-2012004567-A2 FLUORINE RADIOLABELLING PROCESS ISIS INNOVATION LIMITED (GB) 2012-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130190529-A1 Fluorine Radiolabelling Process ESRRG, NR5A2, RXFP4 ESR1 78/4885GRIN1 1456/4885GRIN2B 1379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.