Benzene

Benzene

SCHEMBL3268864

COC(=O)C1=C(C)NC(COCCN)=C(C(=O)O)C1c1ccccc1Cl.c1ccccc1

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 4/20 0.82
ADORA3 P0DMS8 4/20 0.82
TBXA2R P21731 3/20 0.82
ADRA1A P35348 3/20 0.82
SLC6A3 Q01959 3/20 0.82
DRD1 P21728 3/20 0.82
OPRM1 P35372 3/20 0.82
KCNH2 Q12809 3/20 0.82
SCN5A Q14524 3/20 0.82
HTR1A P08908 2/20 0.82
ADRA2A P08913 2/20 0.82
CHRM1 P11229 2/20 0.82
SLC6A2 P23975 2/20 0.82
DRD3 P35462 2/20 0.82
ABCB1 P08183 2/20 0.82
ADRB3 P13945 2/20 0.82
OPRK1 P41145 2/20 0.82
KCNK2 O95069 2/20 0.82
HTR2C P28335 2/20 0.82
HTR2B P41595 2/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3183503 1.00 ABCB11 (0.82) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL5477299 0.96 ABCB11 (0.82) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL30471867 0.96 ABCB11 (0.82) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL5477290 0.95 ABCB11 (0.90) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL30958564 0.95 ABCB11 (0.90) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL3181827 0.94 CYP3A4 (0.85) ABCB11ADORA3TBXA2RADRA1ASLC6A3
Benzene SCHEMBL7444141 0.93 TBXA2R (0.70) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL34462108 0.93 TBXA2R (0.70) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL16634960 0.93 TBXA2R (0.70) ABCB11ADORA3TBXA2RADRA1ASLC6A3
SCHEMBL1610044 0.93 TBXA2R (0.70) ABCB11ADORA3TBXA2RADRA1ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132195-A1 ACETONE SOLVATE OF PHTHALOYL AMLODIPINE Esteve Química, S.A. (ES) 2009-12-16 EP claimed
WO-2008119759-A1 ACETONE SOLVATE OF PHTHALOYL AMLODIPINE Esteve Química, S.A. (ES) 2008-10-09 WO claimed
EP-1975167-A1 Acetone solvate of phthaloyl amlodipine ESTEVE QUIMICA, S.A. (ES) 2008-10-01 EP claimed
EP-2132195-B1 ACETONE SOLVATE OF PHTHALOYL AMLODIPINE ESTEVE QUIMICA SA (ES) 2010-06-16 EP disclosed
EP-2132195-A1 ACETONE SOLVATE OF PHTHALOYL AMLODIPINE Esteve Química, S.A. (ES) 2009-12-16 EP disclosed
WO-2008119759-A1 ACETONE SOLVATE OF PHTHALOYL AMLODIPINE Esteve Química, S.A. (ES) 2008-10-09 WO disclosed
EP-1975167-A1 Acetone solvate of phthaloyl amlodipine ESTEVE QUIMICA, S.A. (ES) 2008-10-01 EP disclosed