SCHEMBL327111

SCHEMBL327111

[C-]#[N+]c1ccc(SC)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
CYP1A1 P04798 4/20 0.39
CYP1A2 P05177 4/20 0.39
CYP1B1 Q16678 4/20 0.39
SLC6A4 P31645 8/20 0.37
NOS3 P29474 2/20 0.37
NOS1 P29475 2/20 0.37
FBP1 P09467 1/20 0.36
PLK1 P53350 1/20 0.35
MAOA P21397 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12204626 0.85 SLC6A4 (0.40) ALDH1A1SLC6A4MAOASLC6A2SLC6A3
SCHEMBL83839 0.76 ALDH1A1 (0.58) ALDH1A1CYP1A1CYP1A2CYP1B1SLC6A4
SCHEMBL409015 0.76 HDAC3 (0.32)
SCHEMBL26106467 0.73 ALDH1A1 (0.55) ALDH1A1CYP1A1CYP1A2CYP1B1SLC6A4
SCHEMBL998605 0.69
SCHEMBL11463411 0.69 ALDH1A1 (0.37) ALDH1A1CYP1A1CYP1A2CYP1B1SLC6A4
SCHEMBL2986827 0.67 ALDH1A1 (0.50) ALDH1A1CYP1A1CYP1A2CYP1B1SLC6A4
SCHEMBL10300271 0.67 ALDH1A1 (0.50) ALDH1A1SLC6A4NOS3NOS1PLK1
SCHEMBL7033576 0.67 ALDH1A1 (0.50) ALDH1A1CYP1A1CYP1A2CYP1B1SLC6A4
SCHEMBL10528160 0.67 ALDH1A1 (0.50) ALDH1A1SLC6A4NOS3NOS1PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP disclosed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO disclosed