SCHEMBL3274318

SCHEMBL3274318

COc1ccc(Cn2nc(OC3CCN(CCF)CC3)c3c(Oc4ccc(NC(=O)c5ccnn(-c6ccc(F)cc6)c5=O)cc4F)ccnc32)cc1.FCCBr

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AXL P30530 20/20 0.50
MERTK Q12866 20/20 0.50
MET P08581 19/20 0.50
TYRO3 Q06418 15/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1944485 0.98 AXL (0.51) AXLMERTKMETTYRO3
SCHEMBL1945962 0.94 AXL (0.51) AXLMERTKMETTYRO3
SCHEMBL1944677 0.92 AXL (0.53) AXLMERTKMETTYRO3
SCHEMBL1945047 0.92 AXL (0.50) AXLMERTKMETTYRO3
SCHEMBL1947699 0.90 AXL (0.52) AXLMERTKMETTYRO3
SCHEMBL1943791 0.89 MET (0.55) AXLMERTKMETTYRO3
SCHEMBL1944232 0.89 AXL (0.53) AXLMERTKMETTYRO3
SCHEMBL1944230 0.89 AXL (0.53) AXLMERTKMETTYRO3
SCHEMBL3104410 0.88 AXL (0.59) AXLMERTKMETTYRO3
SCHEMBL1945115 0.88 AXL (0.51) AXLMERTKMETTYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193130-A1 PYRAZOLO-PYRIDINES AS TYROSINE KINASE INHIBITORS Array Biopharma, Inc. (US) 2010-06-09 EP disclosed
WO-2009033084-A1 PYRAZOLO-PYRIDINES AS TYROSINE KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2009-03-12 WO disclosed