SCHEMBL3276590

SCHEMBL3276590

Cc1ncnc(C)c1C(=O)N1CC2CN(CCC3(c4cccc(F)c4)CCN(C(=O)O)CC3)CC2C1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 18/20 0.83
CCL5 P13501 4/20 0.55
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3272887 0.93 CCR5 (0.83) CCR5CCL5KCNH2
SCHEMBL3271289 0.93 CCR5 (0.80) CCR5CCL5KCNH2
SCHEMBL3271209 0.91 CCR5 (0.80) CCR5CCL5KCNH2
SCHEMBL3270269 0.91 CCR5 (0.80) CCR5CCL5KCNH2
SCHEMBL3271641 0.91 CCR5 (1.00) CCR5CCL5KCNH2
SCHEMBL3271875 0.91 CCR5 (1.00) CCR5CCL5KCNH2
SCHEMBL3273285 0.90 CCR5 (0.77) CCR5CCL5
SCHEMBL3273108 0.90 CCR5 (0.81) CCR5CCL5KCNH2
SCHEMBL3274753 0.90 CCR5 (0.88) CCR5CCL5KCNH2
SCHEMBL3273167 0.90 CCR5 (1.00) CCR5CCL5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066674-B1 OCTAHYDROPYRROLO [3, 4-C] PYRROLE DERIVATIVES AND THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2010-06-30 EP claimed