SCHEMBL3277339

SCHEMBL3277339

COCCCN1CCOc2ccc(COC3CNCC(O)C3c3ccc(Oc4ccc(C)cc4)cc3)cc21

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
REN P00797 13/20 0.42
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
THRB P10828 1/20 0.32
CYP2C19 P33261 1/20 0.32
TSHR P16473 1/20 0.32
AXL P30530 1/20 0.30
MERTK Q12866 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13161136 1.00 REN (0.42) RENALDH1A1CYP3A4CYP2D6THRB
SCHEMBL3277251 0.95 REN (0.45) RENTSHR
SCHEMBL8435065 0.95 REN (0.43) RENALDH1A1CYP3A4CYP2D6THRB
SCHEMBL13161210 0.95 REN (0.45) RENTSHR
SCHEMBL3267579 0.95 REN (0.43) RENALDH1A1CYP3A4CYP2D6THRB
SCHEMBL8428938 0.94 REN (0.48) RENTSHRAXLMERTK
SCHEMBL4583046 0.94 REN (0.42) RENAXLMERTK
SCHEMBL8430160 0.94 REN (0.49) REN
SCHEMBL8427519 0.94 REN (0.42) RENAXLMERTK
SCHEMBL3272419 0.94 REN (0.48) RENTSHRAXLMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863802-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2010-06-16 EP disclosed
EP-1987834-A2 Substituted piperidines as therapeutic compounds Speedel Experimenta AG (CH) 2008-11-05 EP disclosed