SCHEMBL328273

SCHEMBL328273

C=C(c1ccc(Nc2nc(C)c(CC)nc2C(N)=O)cc1C(F)(F)F)N1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 12/20 0.47
EML4 Q9HC35 11/20 0.47
RET P07949 5/20 0.44
ROS1 P08922 5/20 0.44
FLT3 P36888 5/20 0.44
AXL P30530 4/20 0.40
ETV6 P41212 3/20 0.40
EGFR P00533 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10156548 0.82 ALK (0.48) ALKEML4RETROS1FLT3
SCHEMBL17340282 0.80 ALK (0.46) ALKEML4RETROS1FLT3
SCHEMBL10156818 0.77 ALK (0.70) ALKEML4RETROS1FLT3
SCHEMBL10156944 0.75 ALK (0.60) ALKEML4RETROS1FLT3
SCHEMBL10157381 0.75 ALK (0.60) ALKEML4RETROS1FLT3
SCHEMBL10126641 0.72 EML4 (0.45) ALKEML4RETROS1FLT3
SCHEMBL10155933 0.72 ALK (0.46) ALKEML4RETROS1FLT3
SCHEMBL10156483 0.69 EML4 (0.42) ALKEML4RETROS1FLT3
SCHEMBL10158010 0.68 ALK (0.71) ALKEML4RETROS1FLT3
SCHEMBL10156754 0.68 ALK (0.54) ALKEML4RETROS1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428508-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2012-03-14 EP disclosed