SCHEMBL3284696

SCHEMBL3284696

O=C1Nc2ccccc2C1=Cc1cc2cccccc-2c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 3/20 0.66
RAF1 P04049 2/20 0.65
PDGFRB P09619 4/20 0.63
PLK4 O00444 2/20 0.63
PLK1 P53350 2/20 0.63
RET P07949 1/20 0.63
KDR P35968 1/20 0.63
PIM1 P11309 1/20 0.62
EGFR P00533 3/20 0.60
ERBB2 P04626 3/20 0.60
IGF1R P08069 3/20 0.60
NOX4 Q9NPH5 1/20 0.60
DHFR P00374 1/20 0.60
LRRK2 Q5S007 1/20 0.60
MEN1 O00255 1/20 0.58
NPC1 O15118 1/20 0.58
GMNN O75496 1/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
APP P05067 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13324614 1.00 FLT3 (0.66) FLT3RAF1PDGFRBPLK4PLK1
SCHEMBL3284695 1.00 FLT3 (0.66) FLT3RAF1PDGFRBPLK4PLK1
SCHEMBL16442340 0.87 PDGFRB (0.72) FLT3PDGFRBPLK4PLK1RET
SCHEMBL1301398 0.86 PDGFRB (0.76) FLT3PDGFRBPLK4PLK1RET
SCHEMBL247890 0.86 PDGFRB (0.76) FLT3PDGFRBPLK4PLK1RET
SCHEMBL247891 0.86 PDGFRB (0.76) FLT3PDGFRBPLK4PLK1RET
SCHEMBL29875506 0.86 PDGFRB (0.76) FLT3PDGFRBPLK4PLK1RET
SCHEMBL3283744 0.84 RPS6KA3 (0.66) FLT3RAF1KDRLRRK2MEN1
SCHEMBL3283850 0.84 RPS6KA3 (0.66) FLT3RAF1KDRLRRK2MEN1
SCHEMBL3283740 0.84 RPS6KA3 (0.66) FLT3RAF1KDRLRRK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7714146-B2 Azulene-oxindole compounds as multiple-kinase inhibitors and useful as anticancer agents INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 2010-05-11 US disclosed
US-20080125590-A1 Azulene compounds INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE (TW) 2008-05-29 US disclosed
EP-1918277-A2 Azulene compounds Industrial Technology Research Institute (TW) 2008-05-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080125590-A1 Azulene compounds AZI2, PRMT5, BRCA1 FLT3 796/4885RAF1 1574/4885PDGFRB 671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.