SCHEMBL3289655

SCHEMBL3289655

CCN1C(=O)C(C)(C)Oc2cc(C)c(-c3cc(C=O)ccc3OCC(F)(F)F)cc21

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RXRA P19793 19/20 0.63
DHFR P00374 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3288588 0.89 RXRA (0.78) RXRA
SCHEMBL3291492 0.88 RXRA (0.82) RXRA
SCHEMBL13328323 0.88 RXRA (0.82) RXRA
SCHEMBL3289867 0.87 RXRA (0.62) RXRADHFR
SCHEMBL3288911 0.86 RXRA (0.69) RXRA
SCHEMBL3291223 0.81 RXRA (0.56) RXRA
SCHEMBL3495959 0.79 RXRA (0.80) RXRA
SCHEMBL13328322 0.78 RXRA (1.00) RXRA
SCHEMBL13328327 0.78 RXRA (0.67) RXRA
SCHEMBL3289260 0.78 RXRA (1.00) RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723326-B2 Heterocyclic amide derivatives as RXR agonists for the treatment of dyslipidemia, hypercholesterolemia and diabetes JANSSEN PHARMACEUTICA N.V. (US) 2010-05-25 US disclosed
US-20070078129-A1 Heterocyclic amide derivatives as RXR agonists for the treatment of dyslipidemia, hypercholesterolemia and diabetes JANSSEN PHARMACEUTICA N.V. 2007-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070078129-A1 Heterocyclic amide derivatives as RXR agonists for the treatment of dyslipidemia, hypercholesterolemia and diabetes NR1H2, NR1H3, RXRA RXRA 3/4885DHFR 780/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.