Ipratropium

Ipratropium

SCHEMBL3299299

CC(C)[N+]1(C)[C@@H]2CC[C@H]1CC(OC(=O)C(CO)c1ccccc1)C2.Cl.[Br-]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM3

The experimentally established mechanism targets of Ipratropium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 known ✓ P20309 5/20 0.96
CHRM2 P08172 7/20 0.96
CHRM5 P08912 6/20 0.96
CHRM1 P11229 5/20 0.96
CHRM4 P08173 4/20 0.96
MEN1 O00255 3/20 0.96
KMT2A Q03164 3/20 0.96
SMN1; SMN2 Q16637 2/20 0.96
TSHR P16473 2/20 0.95
BLM P54132 5/20 0.79
PABPC1 P11940 1/20 0.75
CYP2C19 P33261 1/20 0.73
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
HIF1A Q16665 1/20 0.62
HSD17B10 Q99714 1/20 0.62
KDM4E B2RXH2 1/20 0.61
LMNA P02545 1/20 0.61
POLB P06746 1/20 0.61
ADRA2C P18825 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ipratropium SCHEMBL29152427 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL3853 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL3854 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL107906 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL6854302 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL3852 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL16762661 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL6854301 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL30987857 0.99 CHRM2 (0.98) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL99102 0.98 CHRM2 (0.96) CHRM2CHRM5CHRM1CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118126021-A Synthesis method of ipratropium hydrochloride 杭州科巢生物科技有限公司 2024-06-04 CN claimed
EP-3384909-A1 COMBINATION OF OXYMETAZOLINE AND IPRATROPIUM IN TOPICAL NASAL APPLICATION FOR THE TREATMENT OF A COUGH Cortés Borrego, Pablo (MX) 2018-10-10 EP claimed
EP-2170348-B1 EFFERVESCENT TABLETS FOR INHALATORY USE DOMPÉ FARMACEUTICI S P A (IT) 2016-08-10 EP claimed
EP-2978407-A1 AQUEOUS SOLUTION COMPOSITION CONTAINING IPRATROPIUM AND OXYMETAZOLINE Santa Farma Ilaç Sanayi A.S. (TR) 2016-02-03 EP claimed
WO-2014158119-A1 AQUEOUS SOLUTION COMPOSITION CONTAINING IPRATROPIUM AND OXYMETAZOLINE SANTA FARMA İLAÇ SANAYİ A.Ş (TR) 2014-10-02 WO claimed
WO-2014158118-A1 SUSPENSION COMPOSITION CONTAINING IPRATROPIUM AND OXYMETAZOLINE SANTA FARMA İLAÇ SANAYİ A.Ş. (TR) 2014-10-02 WO claimed
US-8450339-B2 Compositions for treatment of common cold TAKEDA PHARMA A/S (DK) 2013-05-28 US claimed
US-20100093783-A1 Composition for treatment of common cold TAKEDA PHARMA A/S (DK) 2010-04-15 US claimed
EP-2170348-A2 EFFERVESCENT TABLETS FOR INHALATORY USE Dompe' S.P.A. (IT) 2010-04-07 EP claimed
WO-2009000473-A2 EFFERVESCENT TABLETS FOR INHALATORY USE DOMPE PHA.R.MA S.P.A. (IT) 2008-12-31 WO claimed
EP-1661570-A2 Compositions comprising ipatropium and xylometazoline for treatment of the common cold Nycomed Danmark ApS (DK) 2006-05-31 EP claimed
EP-1446119-B1 COMPOSITIONS COMPRISING IPATROPIUM AND XYLOMETAZOLINE FOR TREATMENT OF THE COMMON COLD NYCOMED DANMARK APS (DK) 2006-03-01 EP claimed
US-20040248924-A1 Compositions for treatment of common cold TAKEDA PHARMA A/S (DK) 2004-12-09 US claimed
EP-1446119-A2 COMPOSITIONS COMPRISING IPATROPIUM AND XYLOMETAZOLINE FOR TREATMENT OF THE COMMON COLD Nycomed Danmark ApS (DK) 2004-08-18 EP claimed
WO-2003024433-A2 COMPOSITIONS FOR TREATMENT OF COMMON COLD, COMPRISING IPRATROPIUM AND XYLOMETAZOLINE NYCOMED DANMARK APS (DK) 2003-03-27 WO claimed
EP-4642463-A1 PHARMACEUTICAL COMPOSITIONS OF GREEN PROPELLANT Cipla Limited (IN) 2025-11-05 EP disclosed
EP-4323049-B1 UNDERARM SPRAY DELIVERY DEVICE XERO PHARMACEUTICALS IP B V (NL) 2025-05-28 EP disclosed
US-20040248924-A1 Compositions for treatment of common cold TAKEDA PHARMA A/S (DK) 2004-12-09 US disclosed
EP-1446119-A2 COMPOSITIONS COMPRISING IPATROPIUM AND XYLOMETAZOLINE FOR TREATMENT OF THE COMMON COLD Nycomed Danmark ApS (DK) 2004-08-18 EP disclosed
WO-2003024433-A2 COMPOSITIONS FOR TREATMENT OF COMMON COLD, COMPRISING IPRATROPIUM AND XYLOMETAZOLINE NYCOMED DANMARK APS (DK) 2003-03-27 WO disclosed