Edoxaban

Edoxaban

SCHEMBL330046

CN1CCc2nc(C(=O)N[C@@H]3C[C@@H](C(=O)N(C)C)CC[C@@H]3NC(=O)C(=O)Nc3ccc(Cl)cn3)sc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

F10

The experimentally established mechanism targets of Edoxaban. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
F10 known ✓ P00742 20/20 1.00
F2 P00734 2/20 1.00
F5 P12259 1/20 1.00
PLAT P00750 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Edoxaban SCHEMBL716662 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL715418 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL16543780 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL12320151 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL1504007 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL713017 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL715737 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL2125499 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL1312016 1.00 F10 (1.00) F10F2F5PLAT
Edoxaban SCHEMBL715818 1.00 F10 (1.00) F10F2F5PLAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2972 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739305-A1 BUDIODARONE FOR CARDIOVERSION Xyra, LLC (US) 2026-05-13 EP claimed
CN-118108635-B Preparation method of high-purity edoxaban intermediate 广西奕安泰药业有限公司 2026-05-12 CN claimed
US-20260124188-A1 mGluR receptor antagonists for use in prevention andor treatment of bone marrow lesions (BML) andor osteoporosis, cartilage loss, osteosclerosis and osteitis in a mammal ORPHELION AB (SE) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-12605371-B2 Combination therapy for cancer THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-04-21 US claimed
US-20260083773-A1 PEGYLATED MENAQUINOL COMPOSITIONS AND METHODS OF TREATMENT EPIZON PHARMA INC (US) 2026-03-26 US claimed
US-20260071253-A1 METHOD FOR DETECTING THE PRESENCE, IDENTIFICATION AND QUANTIFICATION IN A BLOOD SAMPLE OF ANTICOAGULANTS WHICH ARE BLOOD COAGULATION ENZYMES INHIBITORS, AND MEANS FOR THE IMPLEMENTATION THEREOF STAGO DIAGNOSTICA (FR) 2026-03-12 US claimed
EP-4694945-A1 MEDICAL DEVICES INCLUDING THERAPEUTIC COATINGS FOR LOCAL DELIVERY OF A DIRECT ANTICOAGULANT Boston Scientific Scimed Inc. (US) 2026-02-18 EP claimed
US-12553905-B2 Devices and methods for plasma separation and metering SIEMENS HEALTHCARE DIAGNOSTICS INC. (US) 2026-02-17 US claimed
EP-4438592-B1 EDOXABAN INTERMEDIATE AND PREPARATION METHOD THEREFOR SHANGHAI BIOS TECH CO LTD (CN) 2026-02-11 EP claimed
EP-2383272-A1 ACTIVE BLOOD COAGULATION FACTOR INHIBITOR Daiichi Sankyo Company, Limited (JP) 2011-11-02 EP claimed
US-20110257401-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE CARBOXYLIC ACID DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-10-20 US claimed
EP-2374456-A1 ACTIVATED BLOOD COAGULATION FACTOR X (FXA) INHIBITOR Daiichi Sankyo Company, Limited (JP) 2011-10-12 EP claimed
US-20110077266-A1 Diamine Derivatives DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-03-31 US claimed
US-20100093785-A1 DIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2010-04-15 US claimed
US-20100081685-A1 PHARMACEUTICAL COMPOSITION DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-04-01 US claimed
EP-2140867-A1 PHARMACEUTICAL COMPOSITION Daiichi Sankyo Company, Limited (JP) 2010-01-06 EP claimed
US-20090270446-A1 DIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2009-10-29 US claimed
US-7365205-B2 Cyclic diamine derivatives useful as agents for preventing and/or treating cerebral infarction, cerebral embolism, myocardial infarction, angina pectoris, pulmonary infarction, pulmonary embolism; inhibit activated blood coagulation factor X DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-04-29 US claimed
US-20080015215-A1 DIAMINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2008-01-17 US claimed