SCHEMBL3300938

SCHEMBL3300938

Cc1c(-c2ccccc2)c(N2CC[C@H](N(C)C)C2)c2oc(NCCC(=O)OC(C)(C)C)nc2c1C#N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 5/20 0.33
HRH3 Q9Y5N1 5/20 0.33
HRH4 Q9H3N8 2/20 0.33
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
HTR1D P28221 2/20 0.31
HTR3A P46098 2/20 0.31
HTR6 P50406 2/20 0.31
TMEM97 Q5BJF2 2/20 0.31
USP30 Q70CQ3 2/20 0.31
MAPK8 P45983 2/20 0.31
BTK Q06187 2/20 0.31
MRGPRX2 Q96LB1 2/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3295453 0.93 MCHR1 (0.34) MCHR1HRH3HRH4CTSLCTSB
SCHEMBL3294284 0.91 MCHR1 (0.36) MCHR1HRH3HRH4CTSLCTSB
SCHEMBL3295259 0.88 MCHR1 (0.35) MCHR1HRH3HRH4CTSLCTSB
SCHEMBL3296361 0.88 ELANE (0.41) MCHR1
SCHEMBL3295810 0.82 HTR1D (0.38) MCHR1HRH4HTR1DHTR3AHTR6
SCHEMBL3297029 0.82 HTR1D (0.38) MCHR1HRH4HTR1DHTR3AHTR6
SCHEMBL3296134 0.80 HTR1D (0.35) MCHR1HTR1DHTR3AHTR6TMEM97
SCHEMBL3295465 0.80 HTR1D (0.37) MCHR1HRH3HTR1DHTR3AHTR6
SCHEMBL3295967 0.80 TLR8 (0.34)
SCHEMBL3294683 0.80 NAPEPLD (0.36) MCHR1HRH3CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7737166-B2 Antifungal bicyclic hetero ring compounds DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-06-15 US disclosed
EP-1932837-A1 BICYCLO HETEROCYCLIC COMPOUND HAVING ANTIFUNGAL ACTION Daiichi Sankyo Company, Limited (JP) 2008-06-18 EP disclosed