Chloroquine

Chloroquine

SCHEMBL3302947

CCN(CC)CCCC(C)Nc1ccnc2cc(Cl)ccc12.[PbH2]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.98
CHRM4 P08173 3/20 0.98
CHRM5 P08912 3/20 0.98
ADRA2A P08913 3/20 0.98
CHRM1 P11229 3/20 0.98
ADRA2B P18089 3/20 0.98
ADRA2C P18825 3/20 0.98
CHRM3 P20309 3/20 0.98
KCNH2 Q12809 3/20 0.98
TMEM97 Q5BJF2 2/20 0.98
SIGMAR1 Q99720 2/20 0.98
ACE2 Q9BYF1 2/20 0.98
NR4A2 P43354 2/20 0.98
CYP2D6 P10635 2/20 0.98
PRNP P04156 2/20 0.98
MTOR P42345 2/20 0.98
CYP2C19 P33261 1/20 0.98
TDP1 Q9NUW8 1/20 0.98
APP P05067 1/20 0.98
NQO2 P16083 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R)-Chloroquine SCHEMBL134500 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL8933 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL29363614 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL8934 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL8474661 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
(R)-Chloroquine SCHEMBL29429108 0.99 CHRM2 (1.00) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL23152713 0.98 CHRM2 (0.98) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL5488804 0.98 CHRM2 (0.98) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL9862220 0.98 CHRM2 (0.98) CHRM2CHRM4CHRM5ADRA2ACHRM1
Chloroquine SCHEMBL22534361 0.98 CHRM2 (0.98) CHRM2CHRM4CHRM5ADRA2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2993476-B1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS ENZO LIFE SCIENCES INC (US) 2018-12-26 EP disclosed
EP-3001199-B1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS ENZO LIFE SCIENCES INC (US) 2018-03-21 EP disclosed
EP-3001199-A1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS Enzo Life Sciences, Inc. (US) 2016-03-30 EP disclosed
EP-2499495-B1 Autophagy and phospholipidosis pathway assays ENZO LIFE SCIENCES INC (US) 2016-03-30 EP disclosed
EP-2993476-A1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS Enzo Life Sciences, Inc. (US) 2016-03-09 EP disclosed
EP-2993477-A1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS Enzo Life Sciences, Inc. (US) 2016-03-09 EP disclosed
US-9250249-B2 Autophagy and phospholipidosis pathway assays ENZO BIOCHEM, INC. (US) 2016-02-02 US disclosed
EP-2499495-A1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS Enzo Life Sciences, Inc. (US) 2012-09-19 EP disclosed
WO-2011031330-A1 AUTOPHAGY AND PHOSPHOLIPIDOSIS PATHWAY ASSAYS ENZO LIFE SCIENCES, INC. (US) 2011-03-17 WO disclosed
US-20100093004-A1 Autophagy and phospholipidosis pathway assays ENZO LIFE SCIENCES, INC. 2010-04-15 US disclosed