SCHEMBL3303883

SCHEMBL3303883

CC(C)C[C@H](NC(=O)[C@@H](N)CC(C)C)C(=O)N[C@@H](C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.50
ALDH1A1 P00352 2/20 0.44
BACE1 P56817 2/20 0.44
CTSD P07339 1/20 0.44
FNTA P49354 1/20 0.44
FNTB P49356 1/20 0.44
PGGT1B P53609 1/20 0.44
MAPT P10636 1/20 0.44
LAP3 P28838 3/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
CAPN1 P07384 1/20 0.42
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
ACE P12821 5/20 0.40
LARS1 Q9P2J5 1/20 0.40
MME P08473 1/20 0.40
CPA1 P15085 1/20 0.40
ACE2 Q9BYF1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3303877 1.00 SLC7A5 (0.50) SLC7A5ALDH1A1BACE1CTSDFNTA
SCHEMBL9551440 0.97 SLC7A5 (0.47) SLC7A5ALDH1A1BACE1CTSDFNTA
SCHEMBL10621390 0.97 SLC7A5 (0.47) SLC7A5ALDH1A1BACE1CTSDFNTA
SCHEMBL29591958 0.93 BACE1 (0.47) SLC7A5BACE1CTSDFNTAFNTB
SCHEMBL30753843 0.93 FNTA (0.47) SLC7A5ALDH1A1BACE1CTSDFNTA
SCHEMBL30584447 0.92 BACE1 (0.47) SLC7A5ALDH1A1BACE1CTSDFNTA
Leu-Ala SCHEMBL259115 0.91 SLC7A5 (0.59) SLC7A5ALDH1A1BACE1CTSDMAPT
Leu-Ala SCHEMBL14117889 0.91 SLC7A5 (0.59) SLC7A5ALDH1A1BACE1CTSDMAPT
Leu-Ala SCHEMBL2030930 0.91 SLC7A5 (0.59) SLC7A5ALDH1A1BACE1CTSDMAPT
Leu-Ala SCHEMBL31696288 0.91 SLC7A5 (0.59) SLC7A5ALDH1A1BACE1CTSDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6910 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250206841-A1 ANTI-TROPHOBLAST CELL SURFACE ANTIGEN 2 (TROP-2) ANTIBODIES ADEPT BIOPHARMACEUTICAL AND TECHNOLOGY, LTD. (CN) 2025-06-26 US claimed
CN-119604527-A Anti-programmed death ligand 1 (PD-L1) antibodies 安得泰医药有限公司 2025-03-11 CN claimed
EP-4486783-A2 ANTI-PROGRAMMED DEATH-LIGAND 1 (PD-L1) ANTIBODIES Adept Therapeutics Inc. (US) 2025-01-08 EP claimed
EP-4483959-A2 NOVEL PEPTIDE COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF EYEBIO KOREA (KR) 2025-01-01 EP claimed
CN-118702774-A Preparation method and application of polypeptide coupling compound of targeted GPC-3 protein 上海大学 2024-09-27 CN claimed
US-20240228538-A1 Novel Peptide Compound Or Pharmaceutically Acceptable Salt Thereof EYEBIO KOREA (KR) 2024-07-11 US claimed
US-20240209054-A1 GIP AGONIST COMPOUNDS AND METHODS ZEALAND PHARMA A/S (DK) 2024-06-27 US claimed
CN-117736269-A Polypeptide-photosensitizer targeting GPC-3 as well as preparation method and application thereof 中国人民解放军海军军医大学 2024-03-22 CN claimed
WO-2024059686-A2 DARPIN BACKBONES AND RIGIDIFIED ELECTRON MICROSCOPY IMAGING SCAFFOLDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-03-21 WO claimed
US-20240059753-A1 COMPOSITIONS INCLUDING MULTI-AGONIST PEPTIDES AND METHODS OF MANUFACTURE AND USE PEP2TANGO THERAPEUTICS INC. 2024-02-22 US claimed
EP-4146248-A1 LONG ACTING GLP-1/GIP DUAL AGONISTS Sun Pharmaceutical Industries Limited (IN) 2023-03-15 EP claimed
CN-115768460-A Long-acting GLP-1/GIP dual agonists 太阳医药工业有限公司 2023-03-07 CN claimed
EP-4126920-A2 GIF RECEPTOR AGONIST PEPTIDE COMPOUNDS AND USES THEREOF Takeda Pharmaceutical Company Limited (JP) 2023-02-08 EP claimed
EP-4126921-A2 QD DOSING OF GIP RECEPTOR AGONIST PEPTIDE COMPOUNDS AND USES THEREOF Takeda Pharmaceutical Company Limited (JP) 2023-02-08 EP claimed
WO-2022256800-A2 HUMAN SPERMINE OXIDASE CRYSTAL AND USES THEREOF JANSSEN VACCINES & PREVENTION B.V. (NL) 2022-12-08 WO claimed
CN-115335395-A QD administration of GIP receptor agonist peptide compounds and uses thereof 武田药品工业株式会社 2022-11-11 CN claimed
US-20220227830-A1 QD DOSING OF GIP RECEPTOR AGONIST PEPTIDE COMPOUNDS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-07-21 US claimed
WO-2022148418-A1 PHARMACEUTICAL COMPOSITION CAPABLE OF BEING DELIVERED BY METERED DOSE INHALER 江苏恒瑞医药股份有限公司 2022-07-14 WO claimed
WO-2022079639-A1 GLP-1/GIP DUAL AGONISTS SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2022-04-21 WO claimed
US-20220041676-A1 GIP AGONIST COMPOUNDS AND METHODS ZEALAND PHARMA A/S (DK) 2022-02-10 US claimed