SCHEMBL3310386

SCHEMBL3310386

C=CCCCOC(=O)N[C@@H](CCCC)C(=O)N1C[C@H](OCc2cccc(C=C)c2)C[C@H]1C(=O)OC

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.35
ACE2 Q9BYF1 2/20 0.35
CTSK P43235 3/20 0.34
TGM2 P21980 8/20 0.33
CTSL P07711 2/20 0.33
MC4R P32245 2/20 0.33
MC3R P41968 2/20 0.33
MC1R Q01726 2/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
F13A1 P00488 1/20 0.32
TGM1 P22735 1/20 0.32
ABCB1 P08183 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262939 0.96 ACE (0.38) ACEACE2CTSKTGM2CTSL
SCHEMBL3310782 0.92 TGM2 (0.33) ACEACE2CTSKTGM2CTSL
SCHEMBL3307214 0.87 ACE (0.32) ACEACE2CTSKTGM2CTSL
SCHEMBL3249828 0.78 TGM2 (0.34) ACEACE2CTSKTGM2
SCHEMBL3306727 0.77 ACE (0.34) ACEACE2CTSKTGM2CTSL
SCHEMBL1274270 0.77 P2RY12 (0.35)
SCHEMBL3812802 0.76 ABCB1 (0.46) CTSKCTSLABCB1
SCHEMBL3063867 0.76 ABCB1 (0.46) CTSKCTSLABCB1
SCHEMBL1243502 0.76 CYP3A4 (0.34) CTSK
SCHEMBL2429307 0.76 ABCB1 (0.34) MC4RMC3RMC1RABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9738661-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-22 US disclosed
US-9738661-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-22 US disclosed
US-20150266897-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2015-09-24 US disclosed
US-20150266897-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2015-09-24 US disclosed
US-20100099695-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2010-04-22 US disclosed
US-20100099695-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2010-04-22 US disclosed
US-20100099695-A1 HCV NS3 Protease Inhibitors MSD ITALIA S.R.L. (IT) 2010-04-22 US disclosed
WO-2008057209-A1 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100099695-A1 HCV NS3 Protease Inhibitors HAVCR2, GTF3C3, CTSC ACE 89/4885ACE2 141/4885CTSK 121/4885
US-20150266897-A1 HCV NS3 Protease Inhibitors HAVCR2, GTF3C3, CTSC ACE 89/4885ACE2 141/4885CTSK 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.