SCHEMBL3320027

SCHEMBL3320027

O=C(N[C@H]1CC[C@@H](C(=O)Nc2cccc(-c3ccccc3F)c2)CC1)c1cocn1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.46
MAPK1 P28482 1/20 0.45
MAPT P10636 2/20 0.45
GSK3B P49841 2/20 0.45
F10 P00742 1/20 0.45
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
JAK2 O60674 1/20 0.43
F2R P25116 1/20 0.42
POLB P06746 2/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GRM5 P41594 1/20 0.41
GAA P10253 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3341742 0.84 MAPK1 (0.46) ABL1MAPK1MAPTGSK3BF10
SCHEMBL3327025 0.83 GAA (0.55) ABL1MAPK1MAPTGSK3BF10
SCHEMBL3344983 0.83 ACKR3 (0.47) ABL1MAPK1MAPTGSK3BF10
SCHEMBL3346613 0.74 NPY5R (0.49)
SCHEMBL3333820 0.74 MAPT (0.46) ABL1MAPTGSK3BF10TSHR
SCHEMBL12059120 0.71 POLB (0.51) F10SMN1; SMN2POLBHSD17B10
SCHEMBL3362758 0.70 ABL1 (0.52) ABL1MAPTGSK3BALDH1A1
SCHEMBL3343347 0.70 JAK2 (0.48) ABL1MAPK1HPGDSMN1; SMN2KDM4E
SCHEMBL27769316 0.70 KAT6A (0.55) SMN1; SMN2L3MBTL1GRM5
SCHEMBL12058665 0.69 PTPN1 (0.53) MAPTSMN1; SMN2POLBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8653125-B2 Cyclohexane derivative having NPY Y5 receptor antagonism SHIONOGI CO., LTD. (JP) 2014-02-18 US disclosed
US-20120004227-A1 CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM SHIONOGI & CO., LTD. (JP) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004227-A1 CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM NPY5R, NPY1R, NPY2R ABL1 1113/4885MAPK1 850/4885MAPT 4378/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.