SCHEMBL3344983

SCHEMBL3344983

O=C(N[C@H]1CC[C@@H](C(=O)Nc2cccc(-c3ccccc3F)c2)CC1)c1cccc(Cl)n1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.47
ABL1 P00519 1/20 0.47
GRM5 P41594 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
JAK2 O60674 1/20 0.44
MAPT P10636 1/20 0.44
GSK3B P49841 1/20 0.44
MAPK1 P28482 1/20 0.44
F10 P00742 1/20 0.43
CNR2 P34972 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3327025 0.83 GAA (0.55) ABL1HPGDSMN1; SMN2JAK2MAPT
SCHEMBL3341742 0.83 MAPK1 (0.46) ACKR3ABL1KDM4EALDH1A1HPGD
SCHEMBL3320027 0.83 ABL1 (0.46) ABL1GRM5KDM4EALDH1A1HPGD
SCHEMBL3367358 0.75 NPY5R (0.47) ACKR3
SCHEMBL7944353 0.74 CNR2 (0.54) ACKR3GRM5CNR2
SCHEMBL3333820 0.72 MAPT (0.46) ACKR3ABL1MAPTGSK3BF10
SCHEMBL12059120 0.72 POLB (0.51) SMN1; SMN2F10
SCHEMBL12058742 0.71 MGLL (0.55) ACKR3SMN1; SMN2
SCHEMBL27769316 0.70 KAT6A (0.55) GRM5SMN1; SMN2
SCHEMBL10190995 0.70 GNRHR (0.43) ACKR3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8653125-B2 Cyclohexane derivative having NPY Y5 receptor antagonism SHIONOGI CO., LTD. (JP) 2014-02-18 US disclosed
US-20120004227-A1 CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM SHIONOGI & CO., LTD. (JP) 2012-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120004227-A1 CYCLOHEXANE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONISM NPY5R, NPY1R, NPY2R ACKR3 159/4885ABL1 1113/4885GRM5 186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.