Meloxicam

Meloxicam

SCHEMBL332632

Cc1cnc(NC(=O)C2=C(O)c3ccccc3S(=O)(=O)N2C)s1.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS2

The experimentally established mechanism targets of Meloxicam. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 4/20 0.98
PTGS1 P23219 4/20 0.98
ABCB11 O95342 1/20 0.98
GLA P06280 1/20 0.98
EDNRA P25101 1/20 0.98
CYP1A2 P05177 2/20 0.76
CYP3A4 P08684 2/20 0.76
CYP2D6 P10635 2/20 0.76
CYP2C9 P11712 2/20 0.76
LMNA P02545 2/20 0.76
PKM P14618 2/20 0.76
THPO P40225 1/20 0.76
PMP22 Q01453 1/20 0.76
AKR1B1 P15121 1/20 0.65
KDM4E B2RXH2 2/20 0.62
USP2 O75604 2/20 0.62
ALOX15 P16050 1/20 0.62
NFKB1 P19838 1/20 0.62
CYP2C19 P33261 1/20 0.62
BLM P54132 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Meloxicam SCHEMBL3576 0.99 PTGS1 (1.00) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL3752395 0.99 PTGS1 (1.00) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL23589638 0.99 PTGS1 (1.00) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL332206 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL20168549 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL20168506 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL3373822 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL20165003 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL2352397 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA
Meloxicam SCHEMBL7898655 0.98 PTGS1 (0.98) PTGS1PTGS2ABCB11GLAEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200078333-A1 Healthier Aging in Domesticated Animals POSTREL RICHARD (US) 2020-03-12 US claimed
CN-109806228-A A kind of solution containing meloxicam liposome 北京泰德制药股份有限公司 2019-05-28 CN claimed
US-20190030044-A1 HUMAN LIFE EXTENSION THERAPY THROUGH MOLECULAR, CELLULAR AND SUBCELLULAR MANAGEMENT OF BIOCHEMICAL REQUIREMENTS OF MITOCHONDRIA AND OF OTHER ORGANELLE PROCESSES ASSOCIATED WITH THE ADVENT OF DISEASE AND/OR AGING POSTREL RICHARD (US) 2019-01-31 US claimed
US-20190029993-A1 QUALITY OF LIFE EXTENSION THERAPIES RELATING TO AGING, FOOD ALLERGIES, PAIN AND REDUCED VIGOR BY MANAGING MOLECULAR, CELLULAR AND SUBCELLULAR BIOCHEMICAL REQUIREMENTS OF MITOCHONDRIA AND OTHER ORGANELLE PROCESSES REVIGORON LLC 2019-01-31 US claimed
WO-2018118197-A1 HEALTHIER AGING IN DOMESTICATED ANIMALS POSTREL RICHARD (US) 2018-06-28 WO claimed
US-20180168932-A1 Meloxicam Dosage Forms APOTEX TECH INC (CA) 2018-06-21 US claimed
US-20130274235-A1 TREATMENT OF MOTOR NEURON DISEASE THE GENERAL HOSPITAL CORPORATION (US) 2013-10-17 US claimed
WO-2012069842-A1 COMBINATION OF A CYSLT1 ANTAGONIST WITH AN ANTI -ARTHRITIC DRUG FOR THE TREATMENT OF ARTHRITIC DISORDER XARAGEN PHARMA LIMITED (GB) 2012-05-31 WO claimed
WO-2012048330-A2 TREATMENT OF MOTOR NEURON DISEASE THE MCLEAN HOSPITAL CORPORATION (US) 2012-04-12 WO claimed
US-20240216295-A1 Anti-Aging Therapy for Humans and Other Mammals POSTREL RICHARD (US) 2024-07-04 US disclosed
US-20230404942-A1 Life Extension and Quality of Life Improvement for Humans POSTREL RICHARD (US) 2023-12-21 US disclosed
CN-111511350-B Compositions for parenteral administration of therapeutic agents 埃皮辛特瑞柯斯公司 2023-10-13 CN disclosed
US-20230114740-A1 Life Extension and Quality of Life Improvement for Humans and Other Mammals POSTREL RICHARD (US) 2023-04-13 US disclosed
CN-112823787-B Injection containing meloxicam and preparation method thereof 北京泰德制药股份有限公司 2023-02-21 CN disclosed
US-20090076019-A1 METHODS FOR TREATING NEUROLOGICAL DISORDERS OR DAMAGE MOUNT SINAI HOSPITAL (CA) 2009-03-19 US disclosed
CN-101090900-A Process for preparation of high-purity meloxicam and meloxicam potassium salt EGYT GYOGYSZERVEGYESZETI GYAR (HU) 2007-12-19 CN disclosed
EP-1828178-A1 PROCESS FOR PREPARATION OF HIGH-PURITY MELOXICAM AND MELOXICAM POTASSIUM SALT EGIS GYOGYSZERGYAR RT. (HU) 2007-09-05 EP disclosed
WO-2006064298-A1 PROCESS FOR PREPARATION OF HIGH-PURITY MELOXICAM AND MELOXICAM POTASSIUM SALT EGIS GYÓGYSZERGYÁR NYRT. (HU) 2006-06-22 WO disclosed
US-6869948-B1 Meloxicam for oral administration BOEHRINGER INGELHEIM PHARMA KG (DE) 2005-03-22 US disclosed
WO-2004062552-A2 PHARMACEUTICAL COMPOSITION CONTAINING A NSAID AND A BENZIMIDAZOLE DERIVATIVE GALEPHAR M/F (BE) 2004-07-29 WO disclosed