SCHEMBL3327449

SCHEMBL3327449

CC(C)N1CCN(C(=O)[C@H]2CC[C@@H](Nc3cccc(Cl)c3)CC2)CC1C

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
EPHX2 P34913 1/20 0.41
GFER P55789 1/20 0.41
MLNR O43193 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ROCK2 O75116 2/20 0.39
CYP3A4 P08684 2/20 0.39
TRPV1 Q8NER1 1/20 0.38
EGFR P00533 1/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PAK1 Q13153 1/20 0.38
LMNA P02545 1/20 0.38
GRM5 P41594 1/20 0.38
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3324461 1.00 ALDH1A1 (0.42) ALDH1A1HPGDTSHREPHX2GFER
SCHEMBL3324458 1.00 ALDH1A1 (0.42) ALDH1A1HPGDTSHREPHX2GFER
SCHEMBL3325327 0.87 POLB (0.44) ALDH1A1GFERKMT2A
SCHEMBL3325385 0.87 POLB (0.44) ALDH1A1GFERKMT2A
SCHEMBL3325323 0.87 POLB (0.44) ALDH1A1GFERKMT2A
SCHEMBL3326029 0.86 GFER (0.50) ALDH1A1TSHREPHX2GFERROCK2
SCHEMBL3326025 0.86 GFER (0.50) ALDH1A1TSHREPHX2GFERROCK2
SCHEMBL3325322 0.84 ALDH1A1 (0.46) ALDH1A1EPHX2KMT2AMEN1CYP3A4
SCHEMBL3326517 0.84 ALDH1A1 (0.46) ALDH1A1EPHX2KMT2AMEN1CYP3A4
SCHEMBL3325324 0.84 ALDH1A1 (0.46) ALDH1A1EPHX2KMT2AMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100120769-A1 CYCLOHEXYL PIPERAZINYL METHANONE DERIVATIVES NETTEKOVEN MATTHIAS 2010-05-13 US disclosed
US-20070167436-A1 Cyclohexyl piperazinyl methanone derivatives HOFFMANN-LA ROCHE INC. 2007-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100120769-A1 CYCLOHEXYL PIPERAZINYL METHANONE DERIVATIVES HRH3, HRH4, HRH1 ALDH1A1 405/4885HPGD 1000/4885TSHR 97/4885
US-20070167436-A1 Cyclohexyl piperazinyl methanone derivatives HRH3, HRH4, HRH1 ALDH1A1 405/4885HPGD 1000/4885TSHR 97/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.