SCHEMBL3343465

SCHEMBL3343465

COC(=O)c1cc(C(=O)OC)cc(-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.50
PDK2 Q15119 8/20 0.47
RBP4 P02753 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
TSHR P16473 1/20 0.44
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43
SCN9A Q15858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LDHA P00338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21609778 0.92 NOTUM (0.57) NOTUMPDK2RBP4SMN1; SMN2TSHR
SCHEMBL7823276 0.88 PDK2 (0.57) NOTUMPDK2RBP4TSHRSCN9A
SCHEMBL21818278 0.88 PPARG (0.46) NOTUMPDK2SMN1; SMN2PPARGPPARA
SCHEMBL7947891 0.85 BACE1 (0.48) SMN1; SMN2ALDH1A1
SCHEMBL28824318 0.80 SCN9A (0.48) PDK2ALDH1A1HPGDPPARGPPARA
SCHEMBL536257 0.79 NOTUM (0.55) NOTUMPDK2RBP4SMN1; SMN2TSHR
SCHEMBL2776641 0.78 NOTUM (0.54) NOTUMPDK2RBP4SMN1; SMN2ALDH1A1
SCHEMBL3903631 0.78 EGFR (0.57) NOTUMPDK2TSHRLDHA
SCHEMBL29630556 0.78 ALDH1A1 (0.51) ALDH1A1HPGDPPARGPPARAFFAR4
SCHEMBL5934523 0.77 PDK2 (0.49) PDK2SMN1; SMN2TSHRPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042030-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2010-04-15 WO disclosed
WO-2010042030-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2010-04-15 WO disclosed
WO-2008119773-A1 AMIDE DERIVATIVES AS INHIBITORS OF ASPARTYL PROTEASES MEDIVIR AB (SE) 2008-10-09 WO disclosed
WO-2008119773-A1 AMIDE DERIVATIVES AS INHIBITORS OF ASPARTYL PROTEASES MEDIVIR AB (SE) 2008-10-09 WO disclosed