SCHEMBL3344549

SCHEMBL3344549

O=c1ccnc(CCc2ccccc2)[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
TAAR1 Q96RJ0 1/20 0.58
DAO P14920 3/20 0.55
GSK3B P49841 2/20 0.52
PDE10A Q9Y233 1/20 0.51
MMP2 P08253 2/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
RNASEH1 O60930 1/20 0.44
BACE1 P56817 1/20 0.44
MMP9 P14780 1/20 0.43
MMP13 P45452 1/20 0.43
GLA P06280 1/20 0.43
GPR84 Q9NQS5 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2284169 0.84 TAAR1 (0.55) MEN1KMT2ASMN1; SMN2TAAR1DAO
SCHEMBL2483213 0.76 PDE3B (0.42) MEN1KMT2ASMN1; SMN2TAAR1DAO
SCHEMBL4016016 0.76 PDE3B (0.51) MEN1KMT2ASMN1; SMN2TAAR1GSK3B
SCHEMBL3639622 0.73 GPR84 (0.51) MEN1KMT2ASMN1; SMN2TAAR1GSK3B
SCHEMBL570036 0.72 TAAR1 (0.69) SMN1; SMN2TAAR1DAOPDE10ANPC1
SCHEMBL791861 0.71 GPR84 (0.54) KMT2AGSK3BGPR84
SCHEMBL12927964 0.71 DAO (0.49) MEN1KMT2ASMN1; SMN2TAAR1DAO
SCHEMBL14486412 0.71 DAO (1.00) DAOPDE10AMMP2RNASEH1MMP9
SCHEMBL10927286 0.71
SCHEMBL14639314 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039922-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed