SCHEMBL3344560

SCHEMBL3344560

C[Sn](C)(C)c1cc(-c2ccccn2)cs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.47
KDM4E B2RXH2 10/20 0.43
LMNA P02545 5/20 0.43
CCR1 P32246 3/20 0.43
CCR5 P51681 3/20 0.43
CCR8 P51685 3/20 0.43
CYP1A2 P05177 2/20 0.43
POLB P06746 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
RAB9A P51151 7/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 2/20 0.42
NPC1 O15118 6/20 0.41
MAPT P10636 4/20 0.41
GLA P06280 1/20 0.41
CYP2A6 P11509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14106734 0.79 PDE10A (0.50) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL3344484 0.75 KDM4E (0.46) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL10160789 0.75 CYP1A2 (0.44) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL12632125 0.75 PDE10A (0.42) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL5356685 0.74 CYP19A1 (0.49) PDE10AKDM4ELMNACCR1CCR5
Hydrochloric Acid SCHEMBL15910677 0.74 PIK3CD (0.45) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL6193707 0.72 CYP2A6 (0.44) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL28534899 0.71 KDM4E (0.42) PDE10AKDM4ELMNACCR1CCR5
SCHEMBL27623963 0.71 KDM4E (0.45) KDM4ELMNACCR1CCR5CCR8
SCHEMBL6851789 0.70 KDM4E (0.41) PDE10AKDM4ELMNACCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039922-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed