SCHEMBL3344660

SCHEMBL3344660

O=c1[nH]c2cnc3cccnc3c2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.39
KDM4E B2RXH2 2/20 0.38
GABRA1 P14867 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37
GABRA2 P47869 2/20 0.37
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
PDE3B Q13370 3/20 0.36
PDE3A Q14432 3/20 0.36
PDE2A O00408 1/20 0.36
GRM4 Q14833 1/20 0.35
HTR1A P08908 1/20 0.35
DAO P14920 1/20 0.35
ATAD2 Q6PL18 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL202937 0.80 KDM4E (0.40) PARP1KDM4EGABRA1GABRG2GABRB3
SCHEMBL1046464 0.76 CDK4 (0.44) PARP1KDM4EGABRA1GABRG2GABRB3
SCHEMBL16748186 0.74 TYRO3 (0.42) KDM4EPDE3BPDE3APDE2AHTR1A
SCHEMBL30846772 0.73 PARP1 (0.42) PARP1KDM4EGABRA1GABRG2GABRB3
SCHEMBL2326520 0.72 PRMT5 (0.41) PARP1KDM4EADORA3ADORA2AADORA1
SCHEMBL660137 0.71 MAPT (0.50) PARP1KDM4EDAOATAD2CDK4
SCHEMBL11623832 0.71 PARP1 (0.41) PARP1KDM4EGABRA1GABRG2GABRB3
SCHEMBL66937 0.69 PARP1 (0.58) PARP1KDM4EADORA3ADORA2AADORA1
SCHEMBL2326516 0.69 ADORA3 (0.45) PARP1GABRA1GABRG2GABRB3GABRA5
Fumaric Acid SCHEMBL18894354 0.67 MAPT (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038165-A1 IMIDAZO[1,5]NAPHTHYRIDINE COMPOUNDS, THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2010-04-08 WO disclosed