SCHEMBL3344839

SCHEMBL3344839

Cc1cc(=O)n2c3c1ccc(=O)n3[C@H](CN1CCC(NC(=O)O)CC1)C2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.38
POLB P06746 2/20 0.35
MAOB P27338 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MCHR1 Q99705 3/20 0.33
KCNH2 Q12809 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
CCR1 P32246 1/20 0.33
CARM1 Q86X55 1/20 0.33
PRMT6 Q96LA8 1/20 0.33
MCHR2 Q969V1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12113978 0.89 KCNA3 (0.42) TOP2A
SCHEMBL3328189 0.84 TOP2A (0.40) TOP2APOLBMCHR1CCR1CARM1
SCHEMBL3323992 0.84 TOP2A (0.40) TOP2APOLBMCHR1CCR1CARM1
SCHEMBL1312328 0.84 TOP2A (0.35) TOP2A
Hydrochloric Acid SCHEMBL1312760 0.83 TOP2A (0.35) TOP2A
SCHEMBL1312958 0.82 TOP2A (0.33) TOP2A
SCHEMBL3327648 0.80 TOP2A (0.53) TOP2APOLBKCNH2CCR1
SCHEMBL3324741 0.78 TOP2A (0.57) TOP2APOLBCYP3A4CYP2C9CYP2C19
SCHEMBL1313181 0.76 TOP2A (0.61) TOP2AKCNH2
SCHEMBL3730946 0.75 CCR1 (0.35) TOP2APOLBMCHR1CCR1CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043714-A1 TRICYCLIC NITROGEN COMPOUNDS USED AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-22 WO disclosed