SCHEMBL3346599

SCHEMBL3346599

Cc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.68
FFAR1 O14842 1/20 0.44
KCNQ3 O43525 3/20 0.41
KCNQ2 O43526 3/20 0.41
KCNQ4 P56696 2/20 0.40
KCNQ5 Q9NR82 2/20 0.40
PDE2A O00408 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ROCK2 O75116 2/20 0.39
MC4R P32245 1/20 0.38
CASR P41180 1/20 0.38
PAX8 Q06710 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346364 1.00 KCNH2 (0.68) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3350659 0.90 KCNH2 (0.68) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL13365111 0.90 KCNH2 (0.68) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3353009 0.89 KCNH2 (0.67) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3346354 0.89 KCNH2 (0.67) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3346321 0.89 KCNH2 (0.77) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3346490 0.87 KCNH2 (0.65) KCNH2PDE2ACYP3A4CYP2D6CYP2C9
SCHEMBL3347903 0.87 KCNH2 (0.67) KCNH2FFAR1KCNQ3KCNQ2KCNQ4
SCHEMBL3346217 0.86 KCNH2 (0.51) KCNH2FFAR1KCNQ3KCNQ2PDE2A
SCHEMBL3353100 0.82 KCNH2 (0.68) KCNH2FFAR1PDE2ACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed