SCHEMBL3353100

SCHEMBL3353100

COc1cc(OC)cc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.68
MC4R P32245 5/20 0.42
ROCK2 O75116 3/20 0.41
PRKG1 Q13976 2/20 0.41
POLB P06746 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
WDR5 P61964 1/20 0.40
CNR1 P21554 1/20 0.39
MC5R P33032 1/20 0.39
MC3R P41968 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
FFAR1 O14842 1/20 0.39
PDE2A O00408 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346490 0.91 KCNH2 (0.65) KCNH2ROCK2PRKG1POLBMEN1
SCHEMBL3346321 0.84 KCNH2 (0.77) KCNH2MC4RLMNACYP3A4CYP2D6
SCHEMBL3347903 0.83 KCNH2 (0.67) KCNH2MC4RROCK2CYP3A4CYP2D6
SCHEMBL3347178 0.82 KCNH2 (0.53) KCNH2ROCK2PRKG1POLBMEN1
SCHEMBL13365111 0.82 KCNH2 (0.68) KCNH2MC4RROCK2CYP3A4CYP2D6
SCHEMBL3346364 0.82 KCNH2 (0.68) KCNH2MC4RROCK2CYP3A4CYP2D6
SCHEMBL3346599 0.82 KCNH2 (0.68) KCNH2MC4RROCK2CYP3A4CYP2D6
SCHEMBL3350659 0.82 KCNH2 (0.68) KCNH2MC4RROCK2CYP3A4CYP2D6
SCHEMBL3346870 0.82 KCNH2 (0.62) KCNH2MC4RKMT2ASMN1; SMN2CYP3A4
SCHEMBL3346354 0.81 KCNH2 (0.67) KCNH2MC4RROCK2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed