SCHEMBL3347137

SCHEMBL3347137

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1cccnc1)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.55
KCNQ3 O43525 2/20 0.53
KCNQ2 O43526 2/20 0.53
KCNH2 Q12809 1/20 0.49
KCNQ4 P56696 1/20 0.48
KCNQ5 Q9NR82 1/20 0.48
ROCK2 O75116 2/20 0.46
CHRNA7 P36544 3/20 0.45
RECQL P46063 1/20 0.44
KCNA5 P22460 3/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365124 1.00 CYP3A4 (0.55) CYP3A4KCNQ3KCNQ2KCNH2KCNQ4
SCHEMBL3346230 0.88 KCNQ3 (0.66) CYP3A4KCNQ3KCNQ2KCNH2KCNQ4
SCHEMBL13365060 0.87 KCNH2 (0.52) CYP3A4KCNQ3KCNQ2KCNH2KCNQ4
SCHEMBL3346905 0.84 KCNH2 (0.49) CYP3A4KCNQ3KCNQ2KCNH2ROCK2
SCHEMBL13365073 0.83 KCNH2 (0.50) CYP3A4KCNQ3KCNQ2KCNH2KCNQ4
SCHEMBL13364979 0.81 KCNH2 (0.58) KCNQ3KCNQ2KCNH2KCNQ4KCNQ5
SCHEMBL3346373 0.81 KCNH2 (0.57) KCNQ3KCNQ2KCNH2KCNQ4KCNQ5
SCHEMBL3346539 0.81 KCNH2 (0.57) KCNQ3KCNQ2KCNH2KCNQ4KCNQ5
SCHEMBL3348192 0.80 KCNH2 (0.57) KCNQ3KCNQ2KCNH2KCNQ4KCNQ5
SCHEMBL3346676 0.80 KCNQ3 (0.53) KCNQ3KCNQ2KCNH2KCNQ4KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed