SCHEMBL3347384

SCHEMBL3347384

O=C(O)N1CCc2nc3ccnn3c(N3CC(OCc4ccccc4)C3)c2CC1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 16/20 0.51
HTR2A P28223 15/20 0.51
HTR2B P41595 15/20 0.51
DPP4 P27487 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSK P43235 1/20 0.34
RPS6KB1 P23443 1/20 0.34
PKLR P30613 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947932 0.89 HTR2C (0.46) HTR2CHTR2AHTR2B
SCHEMBL2573385 0.83 HTR2C (0.73) HTR2CHTR2AHTR2B
SCHEMBL2573429 0.81 HTR2C (0.50) HTR2CHTR2AHTR2B
SCHEMBL10218414 0.79 HTR2C (0.57) HTR2CHTR2AHTR2B
SCHEMBL9947820 0.78 MEN1 (0.54) HTR2CHTR2AHTR2B
SCHEMBL10216877 0.76 HTR2C (0.62) HTR2CHTR2AHTR2B
SCHEMBL2570503 0.73 HTR2C (0.58) HTR2CHTR2AHTR2B
SCHEMBL2569906 0.73 HTR2C (0.44) HTR2CHTR2AHTR2B
SCHEMBL2569904 0.73 HTR2C (0.44) HTR2CHTR2AHTR2B
SCHEMBL2571912 0.73 MEN1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed