SCHEMBL3347538

SCHEMBL3347538

COC(=O)c1cncc(C#C[Si](C)(C)C)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.58
CYP2A6 P11509 1/20 0.43
ALDH1A1 P00352 2/20 0.42
GRM5 P41594 1/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
KDM4E B2RXH2 2/20 0.38
GLRA3 O75311 1/20 0.37
GLRB P48167 1/20 0.37
LMNA P02545 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
MAPT P10636 2/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
S1PR1 P21453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23012593 0.84 ATM (0.57) ATMCYP2A6ALDH1A1GRM5CYP11B1
SCHEMBL28823048 0.84 ATM (0.40) ATMGRM5LMNAMAPTCYP2C9
SCHEMBL1477261 0.84 CYP2C19 (0.57) ATMALDH1A1GRM5LMNACA12
SCHEMBL6844757 0.84 ATM (0.50) ATMCYP2A6ALDH1A1GRM5CYP11B1
SCHEMBL19712252 0.83 KDM4E (0.46) ATMALDH1A1KDM4EGLRA3GLRB
SCHEMBL15400163 0.83 KDM4E (0.46) ATMALDH1A1KDM4EGLRA3GLRB
SCHEMBL27870359 0.81 MKNK1 (0.40) ATMCYP11B1CYP11B2MAPTL3MBTL1
SCHEMBL1477039 0.80 MAPT (0.55) ATMALDH1A1GRM5CYP11B1CYP11B2
SCHEMBL22120719 0.79 ATM (0.51) ATMCYP2A6ALDH1A1GRM5CYP11B1
SCHEMBL30234325 0.79 ATM (0.51) ATMCYP2A6ALDH1A1GRM5CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed
US-5624943-A Pyridine compounds which are useful as leukotriene-B4 -antagonists SCHERING AKTIENGESELLSCHAFT (DE) 1997-04-29 US disclosed
EP-0651745-A1 NEW PYRIDINE DERIVATIVES AS LEUKCOTRIENE B 4? ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1995-05-10 EP disclosed
WO-1994002464-A1 NEW PYRIDINE DERIVATIVES AS LEUKCOTRIENE B4 ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1994-02-03 WO disclosed