SCHEMBL27870359

SCHEMBL27870359

C[Si](C)(C)C#Cc1cncc(C(N)=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 4/20 0.40
MKNK2 Q9HBH9 4/20 0.40
SIRT2 Q8IXJ6 4/20 0.39
SIRT1 Q96EB6 4/20 0.39
SIRT3 Q9NTG7 4/20 0.39
RAF1 P04049 1/20 0.38
PKMYT1 Q99640 1/20 0.38
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
F7 P08709 1/20 0.37
F3 P13726 1/20 0.37
SARM1 Q6SZW1 1/20 0.37
SIRT6 Q8N6T7 1/20 0.37
SIRT5 Q9NXA8 1/20 0.37
SIRT4 Q9Y6E7 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DYRK1A Q13627 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347538 0.81 ATM (0.58) CYP11B2CYP11B1L3MBTL1MAPTATM
SCHEMBL28823048 0.80 ATM (0.40) HCAR2NPC1RAB9AL3MBTL1DYRK1A
SCHEMBL22531723 0.78 GRM5 (0.38)
SCHEMBL1477261 0.77 CYP2C19 (0.57) L3MBTL1MAPTATM
SCHEMBL12478968 0.77 GRM5 (0.55) L3MBTL1NNMTMAPT
SCHEMBL1479638 0.77 GRM5 (0.56) MKNK1MKNK2SIRT2SIRT1SIRT3
Hydrochloric Acid SCHEMBL1476861 0.75 GRM5 (0.55) MKNK1MKNK2SIRT2SIRT1SIRT3
SCHEMBL25093690 0.75 NOS1 (0.44) MKNK1MKNK2L3MBTL1NNMTMAPT
SCHEMBL3821120 0.75 CYP11B2 (0.50) MKNK1MKNK2SIRT2SIRT1SIRT3
SCHEMBL28776945 0.75 PARP1 (0.43) MKNK1MKNK2SIRT2SIRT1SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102665718-A Heterocyclic compounds useful as pdk1 inhibitors BIOGEN IDEC INC 2012-09-12 CN disclosed