SCHEMBL3348274

SCHEMBL3348274

Cc1nc(-c2ccc(F)cc2)c(C(=O)N2CCOC2CN)s1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 15/20 0.42
HCRTR2 O43614 15/20 0.42
ALDH1A1 P00352 1/20 0.38
PTGS2 P35354 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348271 0.84 HCRTR1 (0.40) HCRTR1HCRTR2ALDH1A1PTGS2
SCHEMBL3343787 0.84 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL2056850 0.80 HCRTR1 (0.40) HCRTR1HCRTR2PTGS2
SCHEMBL3415467 0.78 HCRTR1 (0.43) HCRTR1HCRTR2PTGS2
SCHEMBL3343689 0.75 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL2056852 0.75 HCRTR1 (0.41) HCRTR1HCRTR2PTGS2
SCHEMBL3060001 0.73 HCRTR1 (0.53) HCRTR1HCRTR2ALDH1A1
SCHEMBL3343770 0.73 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL4761846 0.72 PTGS2 (0.54) ALDH1A1PTGS2
SCHEMBL2056960 0.72 HCRTR1 (0.47) HCRTR1HCRTR2ALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO claimed
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO disclosed