SCHEMBL3348839

SCHEMBL3348839

C[Si](C)(C)C#Cc1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 11/20 0.49
SLC6A2 P23975 1/20 0.46
CA12 O43570 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
CA1 P00915 2/20 0.46
CYP1A2 P05177 1/20 0.41
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30808505 1.00 GRM5 (0.49) GRM5SLC6A2CA12CA2CA9
SCHEMBL3614755 0.85 GRM5 (0.39) GRM5CYP1A2
SCHEMBL31286312 0.80 CA12 (0.62) GRM5SLC6A2CA12CA2CA9
SCHEMBL9302636 0.80 CA12 (0.62) GRM5SLC6A2CA12CA2CA9
SCHEMBL852757 0.79 GRM5 (0.43) GRM5CA12CA9CA1
SCHEMBL9082431 0.78 MEN1 (0.36) GRM5SLC6A2CYP1A2
SCHEMBL30293690 0.78 BACE1 (0.41) GRM5SLC6A2
SCHEMBL25693983 0.78 BACE1 (0.41) GRM5SLC6A2
SCHEMBL23867871 0.78 APP (0.50) GRM5CA12CA2CA9CA1
SCHEMBL31349195 0.78 GRM5 (0.56) GRM5CA12CA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102603568-A Fluorine-containing bis-diphenylacetylene liquid crystal compound and preparation method thereof UNIV BEIJING SCIENCE & TECH 2012-07-25 CN disclosed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed