SCHEMBL3350446

SCHEMBL3350446

O=C(NCc1ccccc1)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.79

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.79
MC4R P32245 4/20 0.67
MAOA P21397 2/20 0.55
RORC P51449 1/20 0.48
ALDH1A1 P00352 1/20 0.47
TACR1 P25103 1/20 0.46
KDM1A O60341 1/20 0.46
MAOB P27338 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365061 1.00 KCNH2 (0.79) KCNH2MC4RMAOARORCALDH1A1
SCHEMBL3346236 0.88 MC4R (0.65) KCNH2MC4RMAOAKDM1ACYP3A4
SCHEMBL23951395 0.87 MC4R (0.77) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL13364991 0.87 MC4R (0.77) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL23951303 0.87 MC4R (0.77) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL3353248 0.86 MC4R (0.68) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL13365063 0.86 MC4R (0.68) KCNH2MC4RALDH1A1TSHRHSD17B10
Hydrochloric Acid SCHEMBL23923790 0.86 MC4R (0.75) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL2226816 0.84 MC4R (0.68) KCNH2MC4RALDH1A1TSHRHSD17B10
SCHEMBL13365062 0.83 KCNH2 (0.57) KCNH2MC4RMAOATACR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed