Cholesterol

Cholesterol

SCHEMBL335591

CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C.[C]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OSBP P22059 6/20 0.98
RORC P51449 5/20 0.98
OSBP2 Q969R2 3/20 0.98
USP2 O75604 1/20 0.98
LMNA P02545 1/20 0.98
ABCB1 P08183 1/20 0.98
CYP46A1 Q9Y6A2 1/20 0.98
GRIN1 Q05586 6/20 0.83
GRIN2A Q12879 6/20 0.83
NR1H3 Q13133 7/20 0.82
CRYAB P02511 1/20 0.79
HMGCR P04035 1/20 0.79
ITGB3 P05106 1/20 0.79
ITGAV P06756 1/20 0.79
SREBF2 Q12772 1/20 0.79
NPC1L1 Q9UHC9 1/20 0.79
GRIN2B Q13224 5/20 0.78
DHCR24 Q15392 1/20 0.76
EPHA2 P29317 1/20 0.74
NR1H2 P55055 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cholesterol SCHEMBL21707472 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL21447271 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL21340667 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL23761109 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL22225160 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL23579652 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL21539517 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL23365796 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL22095727 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA
Cholesterol SCHEMBL21445079 0.99 OSBP (1.00) OSBPRORCOSBP2USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113135971-A Carbon-losing cholestanal, and preparation method and application thereof 成都贝诺科成生物科技有限公司 2021-07-20 CN claimed
US-9427431-B2 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2016-08-30 US disclosed
EP-1067939-B1 USE OF STEROIDAL ALKALOID DERIVATIVES AS INHIBITORS OF HEDGEHOG PROTEIN SIGNALING PATHWAYS UNIV JOHNS HOPKINS (US) 2015-09-16 EP disclosed
US-20120183603-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO BEACHY PHILIP A (US) 2012-07-19 US disclosed
US-8097632-B2 Blocking hedgehog protein transduction signal passageway using alkaloid steroid JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2012-01-17 US disclosed
US-20100273818-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2010-10-28 US disclosed
US-20080058298-A1 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE 2008-03-06 US disclosed
US-7291626-B1 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto JOHN HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2007-11-06 US disclosed
US-20060142245-A1 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto JOHN HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2006-06-29 US disclosed
US-6867216-B1 Inhibitors of hedgehog signal pathways, compositions and uses related thereto JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2005-03-15 US disclosed
US-20020034725-A1 SENSITIZATION OF CELLS TO RADIATION AND AND CHEMOTHERAPY NATIONAL INSTITUTES OF HEALTH, THE 2002-03-21 US disclosed
US-20020006931-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO THE JOHNS HOPKINS UNIVERSITY 2002-01-17 US disclosed
EP-1067939-A1 USE OF STEROIDAL ALKALOID DERIVATIVES AS INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS The Johns Hopkins University, School of Medicine, Office of Technology Licencing (US) 2001-01-17 EP disclosed
EP-0910385-A4 SENSITIZATION OF CELLS TO RADIATION AND CHEMOTHERAPY UNIV PENNSYLVANIA (US) 1999-12-22 EP disclosed
WO-1999052534-A1 USE OF STEROIDAL ALKALOID DERIVATIVES AS INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 1999-10-21 WO disclosed
EP-0910385-A1 SENSITIZATION OF CELLS TO RADIATION AND CHEMOTHERAPY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1999-04-28 EP disclosed
US-5792657-A Steroid secreting human adrenocortical carcinoma cell lines THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-08-11 US disclosed
WO-1997038697-A1 SENSITIZATION OF CELLS TO RADIATION AND CHEMOTHERAPY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1997-10-23 WO disclosed
EP-0527757-A1 COMPOSITION AND METHODS FOR TREATMENT OF ACNE VULGARIS AND RETARDATION OF AGEING. LEUNG LIT HUNG (HK) 1993-02-24 EP disclosed
WO-1991014431-A1 COMPOSITION AND METHODS FOR TREATMENT OF ACNE VULGARIS AND RETARDATION OF AGEING LEUNG LIT HUNG (HK) 1991-10-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120183603-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO SHH, GLI1, SMO OSBP 643/4885RORC 487/4885OSBP2 911/4885
US-20100273818-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO SHH, GLI1, SMO OSBP 643/4885RORC 487/4885OSBP2 911/4885
US-20020006931-A1 INHIBITORS OF HEDGEHOG SIGNALING PATHWAYS, COMPOSITIONS AND USES RELATED THERETO SHH, SMO, GLI1 OSBP 542/4885RORC 444/4885OSBP2 591/4885
US-20080058298-A1 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto SHH, GLI1, SMO OSBP 551/4885RORC 484/4885OSBP2 753/4885
US-20060142245-A1 Inhibitors of hedgehog signaling pathways, compositions and uses related thereto SHH, GLI1, SMO OSBP 643/4885RORC 487/4885OSBP2 911/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.