SCHEMBL3359889

SCHEMBL3359889

Nc1n[nH]c2ccc(-c3ccccc3)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 14/20 1.00
JAK3 P52333 4/20 0.64
TYK2 P29597 3/20 0.64
JAK1 P23458 1/20 0.64
MKNK1 Q9BUB5 1/20 0.63
GSK3A P49840 3/20 0.58
GSK3B P49841 3/20 0.58
ROCK2 O75116 4/20 0.57
MAP4K4 O95819 4/20 0.57
CDK2 P24941 4/20 0.57
AURKB Q96GD4 4/20 0.57
CLK4 Q9HAZ1 4/20 0.57
PLK4 O00444 3/20 0.57
DAPK3 O43293 3/20 0.57
CDK1 P06493 3/20 0.57
MARK3 P27448 3/20 0.57
CLK2 P49760 3/20 0.57
CDK5 Q00535 3/20 0.57
PRKCD Q05655 3/20 0.57
ROCK1 Q13464 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12907246 1.00 JAK2 (1.00) JAK2JAK3TYK2JAK1MKNK1
SCHEMBL10213929 0.90 JAK2 (0.81) JAK2JAK3TYK2JAK1GSK3A
SCHEMBL12907223 0.87 JAK2 (0.77) JAK2JAK3TYK2JAK1MKNK1
SCHEMBL3361070 0.85 JAK2 (1.00) JAK2JAK3MKNK1GSK3AGSK3B
SCHEMBL12907241 0.85 JAK2 (1.00) JAK2JAK3MKNK1GSK3AGSK3B
SCHEMBL10213905 0.85 JAK2 (0.72) JAK2JAK3TYK2JAK1MKNK1
SCHEMBL12907171 0.84 JAK2 (0.72) JAK2JAK3TYK2JAK1GSK3A
SCHEMBL10213932 0.84 JAK2 (0.72) JAK2JAK3TYK2JAK1GSK3A
SCHEMBL31690865 0.84 JAK2 (1.00) JAK2JAK3TYK2JAK1MKNK1
SCHEMBL12907187 0.84 JAK2 (0.72) JAK2JAK3TYK2JAK1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11446398-B2 Regulated biocircuit systems OBSIDIAN THERAPEUTICS, INC. (US) 2022-09-20 US disclosed
US-20210254056-A1 IDENTIFICATION AND TARGETED MODULATION OF GENE SIGNALING NETWORKS CAMP4 THERAPEUTICS CORPORATION 2021-08-19 US disclosed
US-20190192691-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. 2019-06-27 US disclosed
US-7872039-B2 N-3-chlorobenzyl-3-amino-1H-indazole-5-carboxamide; 3-aminoindazoles; glucocorticoid-depedent kinase (SGK) inhibitors; SGK-induced diseases; diabetes, obesity, metabolic syndrome (dyslipidaemia), systemic and pulmonary hypertonia, cardiovascular diseases and renal diseases, fibrosis; inflammatory agents MERCK PATENT GESELLSCHAFT (DE) 2011-01-18 US disclosed
US-7872039-B2 N-3-chlorobenzyl-3-amino-1H-indazole-5-carboxamide; 3-aminoindazoles; glucocorticoid-depedent kinase (SGK) inhibitors; SGK-induced diseases; diabetes, obesity, metabolic syndrome (dyslipidaemia), systemic and pulmonary hypertonia, cardiovascular diseases and renal diseases, fibrosis; inflammatory agents MERCK PATENT GESELLSCHAFT (DE) 2011-01-18 US disclosed
EP-1638941-B1 INDAZOLE, BENZISOXAZOLE, AND BENZISOTHIAZOLE KINASE INHIBITORS ABBOTT LAB (US) 2010-06-02 EP disclosed
US-20070232620-A1 3-Aminoindazoles MERCK PATENT GMBH (DE) 2007-10-04 US disclosed
US-20070232620-A1 3-Aminoindazoles MERCK PATENT GMBH (DE) 2007-10-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070232620-A1 3-Aminoindazoles SGK3, SGK1, SGK2 JAK2 562/4885JAK3 180/4885TYK2 140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.