SCHEMBL3360704

SCHEMBL3360704

NC1=NCc2cccnc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
ADRA2A P08913 3/20 0.41
ADRA2B P18089 3/20 0.41
ADRA2C P18825 3/20 0.41
HTR5A P47898 5/20 0.37
NOS3 P29474 3/20 0.34
NOS2 P35228 3/20 0.34
TDP2 O95551 2/20 0.34
NSD2 O96028 2/20 0.34
PAX8 Q06710 2/20 0.34
NOS1 P29475 2/20 0.34
ABL1 P00519 1/20 0.34
PLCG1 P19174 1/20 0.34
CES1 P23141 1/20 0.34
RIN1 Q13671 1/20 0.34
MEN1 O00255 1/20 0.34
THRB P10828 1/20 0.34
BLM P54132 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31703946 1.00 TSHR (0.48) TSHRADRA2AADRA2BADRA2CHTR5A
SCHEMBL577689 0.67 TDP1 (0.42) TSHRTDP2NSD2PAX8ABL1
SCHEMBL4095527 0.67 HRH1 (0.49) ADRA2AADRA2BADRA2CTDP2NSD2
SCHEMBL1194687 0.67 TSHR (0.95) TSHRADRA2AADRA2BADRA2CHTR5A
SCHEMBL31703623 0.67 TSHR (0.95) TSHRADRA2AADRA2BADRA2CHTR5A
SCHEMBL5242604 0.67 HSP90AA1 (0.39) ADRA2AADRA2BADRA2CNOS3NOS2
SCHEMBL7633795 0.67 TSHR (0.48) TSHRNOS3NOS2TDP2NSD2
SCHEMBL1730521 0.65 TSHR (0.38) TSHRHTR5ANOS3NOS2NSD2
Hydrochloric Acid SCHEMBL4092945 0.65 TSHR (1.00) TSHRADRA2AADRA2BADRA2CHTR5A
Hydrochloric Acid SCHEMBL29386664 0.65 TSHR (1.00) TSHRADRA2AADRA2BADRA2CHTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056194-A1 5H-PYRROLO [ 3, 4-B] PYRIDIN DERIVATIVES AND THEIR USE ASTRAZENECA AB (SE) 2010-05-20 WO claimed
WO-2010056194-A1 5H-PYRROLO [ 3, 4-B] PYRIDIN DERIVATIVES AND THEIR USE ASTRAZENECA AB (SE) 2010-05-20 WO disclosed