SCHEMBL3361887

SCHEMBL3361887

CC(C)(C)OC(=O)NC(C(=O)c1nc(C2CC2)sc1-c1ccc(F)cc1)C1CCCCN1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.39
HCRTR2 O43614 5/20 0.39
SCN9A Q15858 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3043816 0.93 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL3002225 0.90 HCRTR1 (0.34) HCRTR1HCRTR2
SCHEMBL3055330 0.87 SCN9A (0.34) HCRTR1HCRTR2SCN9A
SCHEMBL3640420 0.87 SCN9A (0.34) HCRTR1HCRTR2SCN9A
SCHEMBL3363371 0.86 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL3361282 0.86 PTPRB (0.36) HCRTR1HCRTR2SCN9A
SCHEMBL3638060 0.86 PTPRB (0.36) HCRTR1HCRTR2SCN9A
SCHEMBL3365575 0.86 HCRTR1 (0.36) HCRTR1HCRTR2
SCHEMBL3641223 0.85 HCRTR1 (0.38) HCRTR1HCRTR2
SCHEMBL3045164 0.85 HCRTR1 (0.38) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155739-B1 2-CYCLOPROPYL-THIAZOLE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-10-06 EP disclosed