Didanosine

Didanosine

SCHEMBL3363

O=c1[nH]cnc2c1ncn2[C@H]1CC[C@@H](CO)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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The experimentally established mechanism targets of Didanosine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 1.00
LMNA P02545 1/20 1.00
ALB P02768 1/20 1.00
MAPK1 P28482 1/20 1.00
TDP1 Q9NUW8 1/20 0.53
CYP1A2 P05177 1/20 0.52
ADORA3 P0DMS8 1/20 0.49
TYMP P19971 2/20 0.48
STING1 Q86WV6 2/20 0.46
P2RX3 P56373 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Didanosine SCHEMBL16695883 1.00 ALDH1A1 (1.00) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL16695888 1.00 ALDH1A1 (1.00) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL16695885 1.00 ALDH1A1 (1.00) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL1674335 1.00 ALDH1A1 (1.00) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL5021456 1.00 ALDH1A1 (1.00) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL7904473 0.98 ALDH1A1 (0.95) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL887093 0.95 ALDH1A1 (0.91) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL284944 0.95 ALDH1A1 (0.91) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL2327408 0.92 ALDH1A1 (0.85) ALDH1A1LMNAALBMAPK1TDP1
Didanosine SCHEMBL7787270 0.92 ALDH1A1 (0.84) ALDH1A1LMNAALBMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 43421 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2026-05-28 US claimed
EP-4746907-A1 METHOD OF TREATMENT OF HIV INFECTION WITH VACCINE Gilead Sciences, Inc. (US) 2026-05-27 EP claimed
WO-2026104544-A1 EXO-VINYLENE CARBONATE COMPOUNDS AS PRECURSORS FOR ISOCYANATE-FREE URETHANE-TYPE POLYMERS BASF SE (DE) 2026-05-21 WO claimed
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
EP-4745170-A1 METHOD FOR PREPARING A URETHANE GROUP-CONTAINING POLYMER BASF SE (DE) 2026-05-20 EP claimed
EP-4094767-B1 NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO UNIV EMORY (US) 2026-05-20 EP claimed
EP-4745169-A1 COMPOSITION USEFUL AS COATING, SEALANT OR ADHESIVE BASF SE (DE) 2026-05-20 EP claimed
US-20260124290-A1 HIV Immunogens, Vaccines, and Methods Related Thereto UNIV EMORY (US) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
WO-2026085583-A1 MOLECULAR ASSAY FOR DETECTING HIV-1 DRUG-RESISTANT MUTATIONS ST VINCENT'S HOSPITAL SYDNEY LIMITED (AU) 2026-04-30 WO claimed
WO-1991018089-A1 ASSOCIATION BETWEEN A HUMAN IMMUNODEFICIENCY VIRUS-RELATED RETROVIRUS AND SJOGREN'S SYNDROME GARRY ROBERT F JR (US) 1991-11-28 WO claimed
WO-1991013623-A1 C-5 MONO-SUBSTITUTED BARBITURATES IN COMBINATION WITH THERAPEUTIC AGENTS AND USES THEREOF MEMORIAL HOSPITAL FOR CANCER AND ALLIED DISEASES (US) 1991-09-19 WO claimed
WO-1991009605-A1 TREATMENT OF HUMAN RETROVIRAL INFECTIONS WITH 2',3'-DIDEOXYINOSINE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1991-07-11 WO claimed
EP-0416011-A4 CHEMOTHERAPEUTIC COMPOSITION FOR AIDS US COMMERCE (US) 1991-05-22 EP claimed
EP-0416011-A1 CHEMOTHERAPEUTIC COMPOSITION FOR AIDS THE UNITED STATES OF AMERICA as represented by the Secretary United States Department of Commerce (US) 1991-03-13 EP claimed
EP-0398230-A2 Antiviral, highly water soluble, stable, crystalline salts of 2',3'-dideoxyinoside monohydrate, 2',3'-dideoxy-2',3'-didehydrothymidine monohydrate and 2',3'-dideoxy-2'-fluoroinosine hemihydrate Bristol-Myers Squibb Company (US) 1990-11-22 EP claimed
WO-1990011081-A1 INHIBITION OF HIV USING SYNERGISTIC COMBINATIONS OF NUCLEOSIDE DERIVATIVES ONCOGEN LIMITED PARTNERSHIP (US) 1990-10-04 WO claimed
WO-1989011277-A2 PORPHYRIN AND PHTHALOCYANINE ANTIVIRAL COMPOSITIONS GEORGIA STATE UNIVERSITY FOUNDATION, INC. (US) 1989-11-30 WO claimed
WO-1989011274-A1 CHEMOTHERAPEUTIC COMPOSITION FOR AIDS THE UNITED STATES OF AMERICA, AS REPRESENTED BY TH (US) 1989-11-30 WO claimed
WO-1987001284-A1 INHIBITION OF IN VITRO INFECTIVITY AND CYTOPATHIC EFFECT OF HTLV-III/LAV BY 2',3'-DIDEOXYNOSINE, 2',3'-DIDEOXYGUANOSINE, OR 2',3'-DIDEOXYADENOSINE UNITED STATES OF AMERICA, REPRESENTED BY THE UNITE (US) 1987-03-12 WO claimed