SCHEMBL3364860

SCHEMBL3364860

CCOC(=O)N1CC2(CCCNC2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.51
OPRM1 P35372 1/20 0.38
LMNA P02545 2/20 0.37
NLRP3 Q96P20 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 1/20 0.36
BCHE P06276 1/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
AKT1 P31749 1/20 0.35
ADORA1 P30542 1/20 0.35
APP P05067 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6543487 0.85 NOTUM (0.55) NOTUMOPRM1BCHEGAASMN1; SMN2
SCHEMBL3363958 0.85 NOTUM (0.50) NOTUMBCHEROCK2ROCK1HDAC1
SCHEMBL28312084 0.76 SLC18A3 (0.46) NOTUMALDH1A1SMN1; SMN2HDAC1HDAC8
SCHEMBL6544398 0.73 NPC1 (0.51) NOTUML3MBTL1GAASMN1; SMN2AKT1
SCHEMBL14529913 0.73 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1HDAC1
Hydrochloric Acid SCHEMBL7565105 0.72 NPC1 (0.50) NOTUML3MBTL1GAASMN1; SMN2AKT1
SCHEMBL14530335 0.72 HDAC1 (0.59) NOTUML3MBTL1ALDH1A1GAASMN1; SMN2
SCHEMBL29644467 0.70 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1HDAC1
SCHEMBL6543338 0.70 NOTUM (0.57) NOTUMAKT1ROCK2ROCK1HDAC1
Hydrochloric Acid SCHEMBL7497468 0.70 NOTUM (0.39) NOTUMALDH1A1SMN1; SMN2AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996590-B1 SPIROINDOLINONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-10-06 EP disclosed
EP-1996590-A1 SPIROINDOLINONE DERIVATIVES F. Hoffmann-la Roche AG (CH) 2008-12-03 EP disclosed
WO-2007104664-A1 SPIROINDOLINONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-09-20 WO disclosed