SCHEMBL3363958

SCHEMBL3363958

CC(C)(C)OC(=O)N1CC2(CCCNC2)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.50
KDM1A O60341 1/20 0.49
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC8 Q9BY41 2/20 0.40
BCHE P06276 1/20 0.37
MAPK1 P28482 1/20 0.35
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
PDK2 Q15119 1/20 0.34
CYP11B2 P19099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1222469 0.86 NOTUM (0.53) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL30413026 0.86 NOTUM (0.53) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL3364860 0.85 NOTUM (0.51) NOTUMHDAC1HDAC6HDAC8BCHE
Hydrochloric Acid SCHEMBL25232027 0.85 NOTUM (0.52) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL17807330 0.84 NOTUM (0.64) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL13085702 0.79 KDM1A (0.56) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL29384374 0.79 KDM1A (0.56) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL25350959 0.79 NOTUM (0.53) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL30898670 0.79 NOTUM (0.53) NOTUMKDM1AHDAC1HDAC6HDAC8
SCHEMBL15676941 0.79 NOTUM (0.53) NOTUMKDM1AHDAC1HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996590-B1 SPIROINDOLINONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-10-06 EP disclosed