SCHEMBL3365373

SCHEMBL3365373

Cn1nc2c(-c3ccc(Cl)cc3Cl)cccc2c1CNC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 10/20 0.46
CNR1 P21554 8/20 0.44
P2RX7 Q99572 1/20 0.39
SHMT1 P34896 1/20 0.39
SHMT2 P34897 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366146 0.89 CRHR1 (0.43) CRHR1CNR1P2RX7SHMT1SHMT2
Hydrochloric Acid SCHEMBL3366143 0.89 CRHR1 (0.43) CRHR1CNR1P2RX7SHMT1SHMT2
SCHEMBL3364385 0.89 CRHR1 (0.41) CRHR1CNR1P2RX7
SCHEMBL3364388 0.85 CRHR1 (0.48) CRHR1
Hydrochloric Acid SCHEMBL3365148 0.84 CRHR1 (0.47) CRHR1
SCHEMBL3363727 0.84 CRHR1 (0.47) CRHR1
SCHEMBL14206651 0.83 MAPK8 (0.43) CNR1
Hydrochloric Acid SCHEMBL3362608 0.83 CRHR1 (0.46) CRHR1
SCHEMBL3364574 0.83 CRHR1 (0.50) CRHR1
SCHEMBL3839128 0.81 CRHR1 (0.51) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed