SCHEMBL3366528

SCHEMBL3366528

O=C(c1c(F)c(F)c(F)c(F)c1F)N1CCCC1c1nnc(-c2ccc(-c3ccccc3)cc2)o1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 15/20 0.57
HCRTR2 O43614 14/20 0.57
USP30 Q70CQ3 1/20 0.48
DPP4 P27487 1/20 0.48
HSD11B1 P28845 1/20 0.44
NPC1 O15118 1/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 1/20 0.44
HDAC3 O15379 1/20 0.43
CYP2C9 P11712 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366901 0.87 HCRTR1 (0.61) HCRTR1HCRTR2USP30DPP4HSD11B1
SCHEMBL3366778 0.85 HCRTR1 (0.58) HCRTR1HCRTR2USP30DPP4HSD11B1
SCHEMBL3367428 0.85 HCRTR1 (0.55) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL3367310 0.84 HCRTR1 (0.61) HCRTR1HCRTR2HSD11B1
SCHEMBL3369211 0.83 HCRTR1 (0.60) HCRTR1HCRTR2USP30DPP4HSD11B1
SCHEMBL3370370 0.83 HCRTR1 (0.60) HCRTR1HCRTR2USP30DPP4HSD11B1
SCHEMBL3366195 0.82 HCRTR1 (0.56) HCRTR1HCRTR2USP30HSD11B1NPC1
SCHEMBL3370194 0.81 GRM5 (0.60) HCRTR1HCRTR2USP30DPP4
SCHEMBL3369475 0.81 HCRTR1 (0.61) HCRTR1HCRTR2USP30DPP4HSD11B1
SCHEMBL3368643 0.80 HCRTR1 (0.53) HCRTR1HCRTR2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed