SCHEMBL3367002

SCHEMBL3367002

CC1=NNC(=O)C1=Cc1ccc(-c2cccc(C(=O)N3CCCN(C)CC3)c2)o1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 11/20 0.67
PIM2 Q9P1W9 9/20 0.67
FLT3 P36888 2/20 0.67
PIM3 Q86V86 1/20 0.67
MEN1 O00255 2/20 0.45
POLB P06746 2/20 0.45
KMT2A Q03164 2/20 0.45
GFER P55789 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
PSMD14 O00487 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MMP2 P08253 1/20 0.43
MAPT P10636 1/20 0.43
DNMT1 P26358 1/20 0.43
RECQL P46063 1/20 0.43
MCL1 Q07820 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
BRAF P15056 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366998 1.00 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL12989976 1.00 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL31434359 0.85 PIM1 (0.82) PIM1PIM2FLT3PIM3MEN1
SCHEMBL31434336 0.83 PIM1 (0.84) PIM1PIM2FLT3PIM3ALDH1A1
SCHEMBL12990510 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL3363073 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL3363071 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL3363065 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL12990513 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1
SCHEMBL3363075 0.82 PIM1 (0.67) PIM1PIM2FLT3PIM3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100331315-A1 RHODANINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS SENHWA BIOSCIENCES, INC. (TW) 2010-12-30 US disclosed
WO-2010148351-A1 RHODANINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS CYLENE PHARMACEUTICALS, INC. (US) 2010-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331315-A1 RHODANINES AND RELATED HETEROCYCLES AS KINASE INHIBITORS PIM2, PIM1, CDK2 PIM1 2/4885PIM2 1/4885FLT3 90/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.