SCHEMBL3367409

SCHEMBL3367409

CC(c1ccccc1)N1c2nc(-c3ccncn3)cc(=O)n2CCC12CCCC2

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.47
CYP2D6 P10635 5/20 0.45
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370809 0.98 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3369881 0.86 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3364467 0.84 GSK3B (0.42) GSK3BCYP2D6CYP1A2
SCHEMBL3364472 0.83 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3366174 0.82 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3364868 0.82 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3366183 0.82 GSK3B (0.51) GSK3BCYP2D6CYP1A2
SCHEMBL3367413 0.81 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3364483 0.81 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3366617 0.81 GSK3B (0.43) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603915-B1 SUBSTITUTED 8 -PYRIDINYL-DIHYDROSPIRO- CYCLOALKYL -PYRIMIDO 1,2-a PYRIMIDIN-6-ONE AND 8 -PYRIMIDIN YL-DIHYDROSPIRO- CYCLOALKYL -PYRIMIDO 1,2-a PYRIMIDIN-6-ONE DERIVATIVES AND THEIR USE AGAINST NEUROGENERATIVE DISEASES SANOFI AVENTIS (FR) 2010-05-26 EP claimed