SCHEMBL3368321

SCHEMBL3368321

N#CC1(c2ccc(-c3ccc(N4C[C@H](Cn5ccnn5)OC4=O)cc3)cc2F)C2CNCC21

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 16/20 0.55
KCNH2 Q12809 1/20 0.51
CYP3A4 P08684 3/20 0.51
MAOB P27338 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13334899 1.00 MAOA (0.55) MAOAKCNH2CYP3A4MAOBCYP2D6
Hydrochloric Acid SCHEMBL3371870 0.99 MAOA (0.54) MAOAKCNH2CYP3A4MAOBCYP2D6
SCHEMBL13334916 0.93 MAOA (0.54) MAOAKCNH2CYP3A4MAOBCYP2D6
SCHEMBL13335196 0.93 MAOA (0.62) MAOAKCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL3368921 0.93 MAOA (0.62) MAOAKCNH2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL3368091 0.92 MAOA (0.54) MAOAKCNH2CYP3A4MAOBCYP2D6
Hydrochloric Acid SCHEMBL3366681 0.92 MAOA (0.61) MAOAKCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL5789875 0.85 KCNH2 (0.50) MAOAKCNH2CYP3A4MAOBCYP2D6
SCHEMBL13335061 0.85 MAOA (0.62) MAOAKCNH2CYP3A4MAOBCYP2D6
SCHEMBL13335259 0.85 MAOA (0.64) MAOAKCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646629-B1 CYCLOPROPYL GROUP SUBSTITUTED OXAZOLIDINONE ANTIBIOTICS AND DERIVATIVES THEREOF MERCK SHARP & DOHME (US) 2010-06-23 EP claimed