SCHEMBL3368865

SCHEMBL3368865

COc1ccc(-c2nccc(NC3=CCOO3)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 9/20 0.52
CLK1 P49759 1/20 0.48
NPC1 O15118 3/20 0.45
DYRK1A Q13627 4/20 0.44
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
MAPT P10636 3/20 0.44
ALDH1A1 P00352 5/20 0.42
LMNA P02545 3/20 0.42
MAPK1 P28482 3/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 6/20 0.40
CYP2D6 P10635 5/20 0.40
USP2 O75604 5/20 0.40
CYP1A2 P05177 5/20 0.40
CYP2C19 P33261 5/20 0.40
TSHR P16473 4/20 0.40
ALOX15 P16050 2/20 0.40
HSD17B10 Q99714 3/20 0.40
CASP7 P55210 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883128 0.83 ABCG2 (0.48) CLK4NPC1DYRK1AMEN1KMT2A
SCHEMBL3368861 0.78 CLK4 (0.52) CLK4CLK1NPC1DYRK1AMEN1
SCHEMBL28233415 0.74 CLK4 (0.67) CLK4CLK1NPC1DYRK1AMEN1
SCHEMBL28294649 0.67 NPC1 (0.87) CLK4CLK1NPC1DYRK1AMEN1
SCHEMBL2666274 0.66 CLK4 (0.63) CLK4CLK1NPC1DYRK1AMEN1
SCHEMBL10505646 0.65 CLK4 (0.61) CLK4CLK1NPC1DYRK1AMEN1
SCHEMBL14679265 0.63 CLK4 (1.00) CLK4NPC1DYRK1AMEN1KMT2A
SCHEMBL28135254 0.63 NPC1 (0.77) CLK4NPC1MEN1KMT2AMAPT
SCHEMBL25002922 0.62 KMT2A (0.56) CLK4CLK1NPC1MEN1KMT2A
SCHEMBL29961676 0.62 NPC1 (0.56) CLK4NPC1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476435-B1 NOVEL PYRIDIN- AND PYRIMIDIN-DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-06-30 EP disclosed