SCHEMBL6883128

SCHEMBL6883128

C1=C(Nc2ccnc(-c3ccccc3)n2)OOC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.48
ITK Q08881 1/20 0.47
CYP1A2 P05177 10/20 0.39
CYP3A4 P08684 10/20 0.39
CYP2D6 P10635 10/20 0.39
CYP2C19 P33261 9/20 0.39
CLK4 Q9HAZ1 9/20 0.39
USP2 O75604 6/20 0.39
MEN1 O00255 6/20 0.39
KMT2A Q03164 6/20 0.39
MAPT P10636 5/20 0.39
KDM4E B2RXH2 3/20 0.39
TSHR P16473 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 1/20 0.37
TP53 P04637 5/20 0.37
ALDH1A1 P00352 5/20 0.37
HSD17B10 Q99714 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3368865 0.83 CLK4 (0.52) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL3370929 0.77 MEN1 (0.43) MEN1KMT2AMAPTKDM4ENPC1
SCHEMBL6883124 0.75 ABCG2 (0.48) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL2422608 0.74 ABCG2 (0.72) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL8346049 0.70 ABCG2 (0.67) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL5261585 0.69 CYP1A2 (0.62) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL11481156 0.68 ADRA2A (0.57) ABCG2ITKCYP2D6CYP2C19MEN1
Hydrochloric Acid SCHEMBL5914224 0.67 CYP1A2 (0.60) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL16926442 0.67 ITK (0.57) ABCG2ITKCYP1A2CYP3A4CYP2D6
SCHEMBL21016714 0.66 ITK (0.52) ABCG2ITKCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068757-A9 NOVEL PYRIDIN- AND PYRIMIDIN-DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-10-07 WO disclosed