SCHEMBL3371353

SCHEMBL3371353

C=C(C(=O)OCC)C(=O)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 1.00
ALDH1A1 P00352 1/20 1.00
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
CES2 O00748 4/20 0.48
CES1 P23141 4/20 0.48
NPC1 O15118 1/20 0.47
EGFR P00533 2/20 0.46
LMNA P02545 2/20 0.46
XBP1 P17861 1/20 0.46
ATM Q13315 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CYP19A1 P11511 2/20 0.44
CASP1 P29466 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97859 0.85 ALDH1A1 (0.73) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
Hydrogen Peroxide SCHEMBL28172477 0.83 ALDH1A1 (0.71) MAPTALDH1A1SMN1; SMN2CES2CES1
Water SCHEMBL27483870 0.83 ALDH1A1 (0.71) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL9578813 0.83 ALDH1A1 (0.71) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL10405628 0.83 ALDH1A1 (0.71) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL27883993 0.83 ALDH1A1 (0.69) MAPTALDH1A1SMN1; SMN2EGFRLMNA
P-Xylene SCHEMBL9441216 0.82 ALDH1A1 (0.68) MAPTALDH1A1MEN1KMT2ACES2
SCHEMBL19626050 0.81 MAPT (0.69) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL316956 0.81 ALDH1A1 (0.69) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL5711212 0.81 ALDH1A1 (0.69) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 119 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363869-B1 PROCESS FOR THE PREPARATION OF ALKYL BENZOYLACRYLATES WEYLCHEM LAMOTTE (FR) 2015-04-08 EP claimed
CN-1243709-C Process for prepn. of alkyl benzoylacrylates CLARIANT FRANCE SA (FR) 2006-03-01 CN claimed
CN-1500074-A Process for prepn. of alkyl benzoylacrylates 克莱里安特法国公司 2004-05-26 CN claimed
EP-1363869-A2 PROCESS FOR THE PREPARATION OF ALKYL BENZOYLACRYLATES Clariant (France) S.A. (FR) 2003-11-26 EP claimed
WO-2002067847-A2 PROCESS FOR THE PREPARATION OF ALKYL BENZOYLACRYLATES CLARIANT (FRANCE) (FR) 2002-09-06 WO claimed
US-4925969-A MICHAEL ADDITION, ALANINE OR LYSINE DERIVATIVE REACTED WITH ETHYL BENZOYLACRYLATE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1990-05-15 US claimed
EP-0052330-B1 NOVEL RESIN COMPOSITION, COATING MATERIAL COMPRISING SAID RESIN COMPOSITION AND METHOD FOR FORMING COATINGS Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-09-05 EP claimed
US-4447580-A POLYMER CONSISTING OF UNSATD AROMATIC AMINE AND UNSATURATED COMPOUND WITH ELECTRON ATTRACTIVE GROUP ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1984-05-08 US claimed
EP-0052330-A1 Novel resin composition, coating material comprising said resin composition and method for forming coatings Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-05-26 EP claimed
JP-61178954-A None JP disclosed
JP-3115254-A None JP disclosed
JP-62129260-A None JP disclosed
CN-114773337-B Method for preparing zolpidem 诚弘制药(威海)有限责任公司 2024-06-21 CN disclosed
CN-116020488-A Preparation method of catalyst for synthesizing lisinopril intermediate 西安凯立新材料股份有限公司 2023-04-28 CN disclosed
US-4562202-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-31 US disclosed
US-4558065-A Derivatives of tricyclic aminoacids, processes for their preparation, agents containing these compounds and their use, and new bicyclic aminoacids as intermediates and processes for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1985-12-10 US disclosed
EP-0052330-B1 NOVEL RESIN COMPOSITION, COATING MATERIAL COMPRISING SAID RESIN COMPOSITION AND METHOD FOR FORMING COATINGS Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-09-05 EP disclosed
US-4447580-A POLYMER CONSISTING OF UNSATD AROMATIC AMINE AND UNSATURATED COMPOUND WITH ELECTRON ATTRACTIVE GROUP ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1984-05-08 US disclosed
US-4442030-A ARALKYLATION WITH BENZOYLACRYLIC ACID, HYDROGENATION, ESTERIFICATION MERCK & CO., INC. (US) 1984-04-10 US disclosed
EP-0052330-A1 Novel resin composition, coating material comprising said resin composition and method for forming coatings Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-05-26 EP disclosed