SCHEMBL3373490

SCHEMBL3373490

NC(=O)c1cccc(C(N)=NO)n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.49
KDM4E B2RXH2 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
ACMSD Q8TDX5 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GNE Q9Y223 1/20 0.36
SCN9A Q15858 1/20 0.35
DGAT1 O75907 1/20 0.35
GAA P10253 1/20 0.34
CYP2C19 P33261 1/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14671991 0.86 KDM4E (0.65) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL2224487 0.86 KDM4E (0.65) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL2224481 0.86 KDM4E (0.65) KDM4EALOX15TSHRACMSDTDP1
Pyridine Dicarboxamide SCHEMBL29587789 0.85 TSHR (0.59) PIM1KDM4EALOX15TSHRACMSD
Pyridine Dicarboxamide SCHEMBL229425 0.85 TSHR (0.59) PIM1KDM4EALOX15TSHRACMSD
Pyridine Dicarboxamide SCHEMBL29501171 0.83 TSHR (0.56) PIM1KDM4EALOX15TSHRACMSD
Pyridine Dicarboxamide SCHEMBL29031925 0.83 TSHR (0.56) PIM1KDM4EALOX15TSHRACMSD
Pyridine Dicarboxamide SCHEMBL15347496 0.83 TSHR (0.56) PIM1KDM4EALOX15TSHRACMSD
Pyridine Dicarboxamide SCHEMBL38659131 0.83 TSHR (0.56) PIM1KDM4EALOX15TSHRACMSD
SCHEMBL20963454 0.80 MAPT (0.50) KDM4ETSHRCYP1A2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1220838-B1 1-AZIRIDINO-1-HYDROXYIMINOMETHYL-DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND MEDICAMENTS CONTAINING SAID COMPOUNDS KALVINS PROF DR IVARS (LV) 2010-11-03 EP disclosed
US-7078418-B1 1-aziridino-1-hydroxyiminomethyl-derivates, method for the production thereof and medicaments containing said compounds Kalvins, Ivars (LV) 2006-07-18 US disclosed